Kinase profiling results of kinases in KIF 2H8HA_H8H (SRC, PDB code: 2H8H, chain A)
Template Kinase: SRC
Template inhibitor: Saracatinib

91 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C C C C C C
PRKCDAGC          
PRKCQAGC          
PKN2AGC          
RPS6KA1AGC          
RPS6KA1CAMK          
RPS6KA2AGC          
RPS6KA2CAMK          
RPS6KA3AGC          
RPS6KA6AGC          
RPS6KA6CAMK          
CHEK1CAMK          
HUNKCAMK          
MGC421053          
NUAK1CAMK          
NUAK2CAMK          
KIAA0999CAMK          
SIK1CAMK          
SIK2CAMK          
MAPK14CMGC          
PLK2Other          
STK36Other          
ULK3Other          
STK39STE          
STK24STE          
MAP2K5STE          
ABL1TK          
ABL2TK          
TNK2TK          
ALKTK          
LTKTK          
CSKTK          
MATKTK          
DDR1TK          
DDR2TK          
EGFRTK          
ERBB2TK          
ERBB3TK          
ERBB4TK          
EPHA1TK          
EPHA3TK          
EPHA4TK          
EPHA5TK          
EPHA6TK          
EPHA8TK          
EPHB1TK          
EPHB2TK          
EPHB3TK          
EPHB4TK          
EPHB6TK          
PTK2BTK          
FERTK          
FESTK          
FGFR1TK          
FGFR2TK          
FGFR3TK          
FGFR4TK          
IGF1RTK          
INSRTK          
INSRRTK          
JAK2TK          
JAK3TK          
TYK2TK          
CSF1RTK          
KITTK          
PDGFRATK          
PDGFRBTK          
RETTK          
FRKTK          
FGRTK          
FYNTK          
SRCTK          
YES1TK          
BLKTK          
HCKTK          
LCKTK          
LYNTK          
PTK6TK          
SRMSTK          
SYKTK          
ZAP70TK          
BMXTK          
BTKTK          
ITKTK          
TECTK          
TXKTK          
NTRK1TK          
NTRK2TK          
NTRK3TK          
IRAK1TKL          
IRAK4TKL          
ACVR1TKL          
ACVRL1TKL          
BMPR1BTKL          

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
PKN2AGC    
PRKCAAGC    
PRKCDAGC    
PRKCQAGC    
RPS6KA1AGC    
RPS6KA2AGC    
RPS6KA3AGC    
RPS6KA6AGC    
CHEK1CAMK    
NUAK1CAMK    
NUAK2CAMK    
SIK2CAMK    
MAPK14CMGC    
PLK2Other    
ULK3Other    
STK24STE    
STK39STE    
ABL1TK    
ABL2TK    
ALKTK    
BLKTK    
BMXTK    
BTKTK    
CSF1RTK    
CSKTK    
DDR2TK    
EGFRTK    
EPHA1TK    
EPHA3TK    
EPHA4TK    
EPHA5TK    
EPHA6TK    
EPHA8TK    
EPHB1TK    
EPHB2TK    
EPHB3TK    
EPHB4TK    
ERBB2TK    
ERBB4TK    
FERTK    
FESTK    
FGFR1TK    
FGFR2TK    
FGFR3TK    
FGFR4TK    
FGRTK    
FRKTK    
FYNTK    
HCKTK    
IGF1RTK    
INSRTK    
INSRRTK    
ITKTK    
JAK2TK    
JAK3TK    
KITTK    
LCKTK    
LTKTK    
LYNTK    
MATKTK    
NTRK1TK    
NTRK2TK    
NTRK3TK    
PDGFRATK    
PDGFRBTK    
PTK2BTK    
PTK6TK    
RETTK    
SRCTK    
SRMSTK    
SYKTK    
TECTK    
TNK2TK    
TXKTK    
TYK2TK    
YES1TK    
ZAP70TK    
ACVR1TKL    
ACVRL1TKL    
IRAK1TKL    
IRAK4TKL