Kinase profiling results of kinases in KIF 2R3OA_2SC (CDK2, PDB code: 2R3O, chain A)
Template Kinase: CDK2
Template inhibitor: 4-(Benzylamino)quinazoline deriv. 28

18 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group
CDK2CMGC
CDK5CMGC
CLK1CMGC
CLK2CMGC
CLK4CMGC
DYRK1ACMGC
DYRK1BCMGC
GSK3BCMGC
MAPK1CMGC
MAPK10CMGC
CHUKOther
ABL1TK
JAK2TK
JAK3TK
METTK
SRCTK
LCKTK

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C
CDC2CMGC  
CDC2CMGC  
CDK2CMGC  
CDK5CMGC  
CLK1CMGC  
CLK2CMGC  
CLK4CMGC  
DYRK1ACMGC  
DYRK1BCMGC  
GSK3BCMGC  
MAPK1CMGC  
MAPK10CMGC  
CHUKOther  
ABL1TK  
JAK2TK  
JAK3TK  
LCKTK  
METTK  
SRCTK