Kinase profiling results of kinases in KIF 3MIYA_B49 (ITK, PDB code: 3MIY, chain A)
Template Kinase: ITK
Template inhibitor: Sunitinib

70 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C
AKT2AGC     
DAPK3CAMK     
CDK2CMGC     
CDK4CMGC     
PCTK2CMGC     
CDK15CMGC     
CDKL2CMGC     
ICKCMGC     
MAKCMGC     
AURKAOther     
AURKBOther     
AURKCOther     
NEK1Other     
DSTYKOther     
TLK2Other     
OXSR1STE     
STK39STE     
STK3STE     
STK4STE     
PAK1STE     
PAK3STE     
TAOK1STE     
TAOK2STE     
TAOK3STE     
STK24STE     
ABL1TK     
TNK1TK     
TNK2TK     
ALKTK     
LTKTK     
MATKTK     
DDR1TK     
DDR2TK     
EGFRTK     
ERBB4TK     
EPHA3TK     
EPHB1TK     
EPHB4TK     
EPHB6TK     
PTK2BTK     
FERTK     
FESTK     
FGFR2TK     
FGFR3TK     
FGFR4TK     
IGF1RTK     
INSRTK     
INSRRTK     
JAK2TK     
METTK     
MUSKTK     
KITTK     
PDGFRATK     
PDGFRBTK     
RETTK     
ROS1TK     
SRCTK     
YES1TK     
BLKTK     
HCKTK     
LCKTK     
BTKTK     
ITKTK     
NTRK1TK     
NTRK2TK     
NTRK3TK     
IRAK4TKL     
RIPK1TKL     

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C C
AKT2AGC      
DAPK3CAMK      
CDC2CMGC      
CDC2CMGC      
CDK2CMGC      
CDK4CMGC      
CDK6CMGC      
CDK6CMGC      
AURKAOther      
AURKBOther      
AURKCOther      
DSTYKOther      
NEK1Other      
TLK2Other      
OXSR1STE      
PAK1STE      
PAK3STE      
STK24STE      
STK3STE      
STK39STE      
STK4STE      
TAOK1STE      
TAOK2STE      
TAOK3STE      
ABL1TK      
ALKTK      
BLKTK      
BTKTK      
DDR2TK      
EGFRTK      
EPHA3TK      
EPHB1TK      
EPHB4TK      
ERBB4TK      
FERTK      
FESTK      
FGFR2TK      
FGFR3TK      
FGFR4TK      
HCKTK      
IGF1RTK      
INSRTK      
INSRRTK      
ITKTK      
JAK2TK      
KITTK      
LCKTK      
LTKTK      
MATKTK      
METTK      
MUSKTK      
NTRK1TK      
NTRK2TK      
NTRK3TK      
PDGFRATK      
PDGFRBTK      
PTK2BTK      
RETTK      
ROS1TK      
SRCTK      
TNK2TK      
YES1TK      
IRAK4TKL