Kinase profiling results of kinases in KIF 2ZM4A_KSM (LCK, PDB code: 2ZM4, chain A)
Template Kinase: LCK
Template inhibitor: BMS-279700

25 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C
CDK2CMGC 
CDK3CMGC 
CDK5CMGC 
MAPK14CMGC 
AURKAOther 
EIF2AK2Other 
PAK4STE 
TNK2TK 
ALKTK 
EGFRTK 
FGFR1TK 
FGFR2TK 
JAK2TK 
PDGFRBTK 
RETTK 
FGRTK 
FYNTK 
SRCTK 
YES1TK 
LCKTK 
NTRK3TK 
IRAK4TKL 
RAF1TKL 

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C
PRKCAAGC   
CDC2CMGC   
CDC2CMGC   
CDK2CMGC   
CDK3CMGC   
CDK5CMGC   
MAPK14CMGC   
AURKAOther   
PAK4STE   
ALKTK   
EGFRTK   
FGFR1TK   
FGFR2TK   
FGRTK   
FYNTK   
JAK2TK   
LCKTK   
NTRK3TK   
PDGFRBTK   
RETTK   
SRCTK   
TNK2TK   
YES1TK   
IRAK4TKL   
RAF1TKL