Kinase profiling results of kinases in KIF 2O0UA_C0M (MAPK10, PDB code: 2O0U, chain A)
Template Kinase: MAPK10
Template inhibitor: ZINC00799686

21 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C
GRK1AGC   
GRK4AGC   
GRK7AGC   
PDPK1AGC   
PRKCQAGC   
SGK3AGC   
PRKD1CAMK   
PRKD2CAMK   
PRKD3CAMK   
CDK2CMGC   
CDKL2CMGC   
DYRK1BCMGC   
HIPK1CMGC   
HIPK2CMGC   
HIPK3CMGC   
HIPK4CMGC   
MAPK10CMGC   
MAPK8CMGC   
MAPK14CMGC   
ICKCMGC   
STK24STE   

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C
GRK4AGC  
GRK7AGC  
PDPK1AGC  
PRKCQAGC  
SGK3AGC  
PRKD1CAMK  
PRKD2CAMK  
PRKD3CAMK  
CDK2CMGC  
DYRK1BCMGC  
HIPK1CMGC  
HIPK2CMGC  
HIPK3CMGC  
HIPK4CMGC  
MAPK10CMGC  
MAPK14CMGC  
MAPK8CMGC  
STK24STE