Kinase profiling results of kinases in KIF 1BL7A_SB4 (MAPK14, PDB code: 1BL7, chain A)
Template Kinase: MAPK14
Template inhibitor: SB220025

22 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group
RPS6KA2AGC
RPS6KA2CAMK
CHEK1CAMK
PRKD3CAMK
CDK2CMGC
CDK3CMGC
CDK5CMGC
CDK9CMGC
CLK2CMGC
GSK3BCMGC
MAPK10CMGC
MAPK8CMGC
MAPK9CMGC
NLKCMGC
MAPK11CMGC
MAPK14CMGC
CHUKOther
FGRTK
FYNTK
SRCTK
YES1TK
LCKTK

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C C
RPS6KA2AGC      
CHEK1CAMK      
PRKD3CAMK      
CDC2CMGC      
CDC2CMGC      
CDK2CMGC      
CDK3CMGC      
CDK5CMGC      
CDK9CMGC      
CLK2CMGC      
GSK3BCMGC      
MAPK10CMGC      
MAPK11CMGC      
MAPK14CMGC      
MAPK8CMGC      
MAPK9CMGC      
NLKCMGC      
CHUKOther      
FGRTK      
FYNTK      
LCKTK      
SRCTK      
YES1TK