Kinase profiling results of kinases in KIF 2JFLA_DKI (SLK, PDB code: 2JFL, chain A)
Template Kinase: SLK
Template inhibitor: 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE

90 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group
CDC42BPB1
DMPKAGC
PDPK1AGC
PRKACAAGC
PRKCDAGC
PRKCQAGC
PRKCEAGC
PKN1AGC
PKN2AGC
RPS6KA4AGC
RPS6KA4CAMK
RPS6KB1AGC
RPS6KA1AGC
RPS6KA1CAMK
RPS6KA2AGC
RPS6KA2CAMK
RPS6KA3AGC
RPS6KA6AGC
RPS6KA6CAMK
CAMK4CAMK
CAMK2BCAMK
CAMK2DCAMK
CAMK2GCAMK
BRSK1CAMK
BRSK2CAMK
MARK2CAMK
MARK4CAMK
NUAK1CAMK
NUAK2CAMK
SIK1CAMK
SIK2CAMK
DAPK3CAMK
STK17ACAMK
DCLK3CAMK
MKNK2CAMK
PHKG1CAMK
PRKD1CAMK
PRKD2CAMK
PRKD3CAMK
CHEK2CAMK
TSSK1BCAMK
CDK2CMGC
CDK3CMGC
CDK5CMGC
CDK9CMGC
CDK11ACMGC
CDK11ACMGC
DYRK1BCMGC
GSK3ACMGC
AURKAOther
AURKBOther
AURKCOther
CAMKK1Other
CAMKK2Other
NEK1Other
NEK3Other
EIF2AK2Other
PLK1Other
PLK3Other
PLK4Other
TLK1Other
TLK2Other
ULK1Other
ULK2Other
PAK4STE
PAK6STE
SLKSTE
STK10STE
STK24STE
STK25STE
ABL1TK
ALKTK
EGFRTK
PTK2TK
FERTK
FESTK
FGFR1TK
FGFR2TK
FGFR3TK
FGFR4TK
IGF1RTK
JAK2TK
JAK3TK
MUSKTK
RETTK
ROS1TK
BMXTK
NTRK1TK
NTRK2TK
NTRK3TK
IRAK4TKL

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C
CDC42BPBAGC  
DMPKAGC  
PDPK1AGC  
PKN1AGC  
PKN2AGC  
PRKACAAGC  
PRKCAAGC  
PRKCDAGC  
PRKCEAGC  
PRKCQAGC  
RPS6KA1AGC  
RPS6KA2AGC  
RPS6KA3AGC  
RPS6KA4AGC  
RPS6KA6AGC  
RPS6KB1AGC  
BRSK1CAMK  
BRSK2CAMK  
CAMK2BCAMK  
CAMK2DCAMK  
CAMK2GCAMK  
CAMK4CAMK  
CHEK2CAMK  
DAPK3CAMK  
MARK2CAMK  
MARK4CAMK  
MKNK2CAMK  
NUAK1CAMK  
NUAK2CAMK  
PHKG1CAMK  
PRKD1CAMK  
PRKD2CAMK  
PRKD3CAMK  
SIK2CAMK  
STK17ACAMK  
TSSK1BCAMK  
CDC2CMGC  
CDC2CMGC  
CDK2CMGC  
CDK3CMGC  
CDK5CMGC  
CDK6CMGC  
CDK6CMGC  
CDK9CMGC  
DYRK1BCMGC  
GSK3ACMGC  
AURKAOther  
AURKBOther  
AURKCOther  
CAMKK1Other  
CAMKK2Other  
NEK1Other  
NEK3Other  
NEK8Other  
PLK1Other  
PLK3Other  
TLK2Other  
ULK1Other  
ULK2Other  
PAK4STE  
PAK6STE  
SLKSTE  
STK10STE  
STK24STE  
STK25STE  
ABL1TK  
ALKTK  
BMXTK  
EGFRTK  
FERTK  
FESTK  
FGFR1TK  
FGFR2TK  
FGFR3TK  
FGFR4TK  
IGF1RTK  
JAK2TK  
JAK3TK  
MUSKTK  
NTRK1TK  
NTRK2TK  
NTRK3TK  
PTK2TK  
RETTK  
ROS1TK  
IRAK4TKL