Kinase profiling results of kinases in KIF 2JDRA_L20 (AKT2, PDB code: 2JDR, chain A)
Template Kinase: AKT2
Template inhibitor: A-443654

44 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C
AKT1AGC 
AKT2AGC 
AKT3AGC 
CITAGC 
ROCK1AGC 
GRK4AGC 
GRK7AGC 
PRKACAAGC 
PRKACBAGC 
PRKXAGC 
PRKCDAGC 
PRKCQAGC 
PRKCEAGC 
PRKCHAGC 
PRKG1AGC 
PRKG2AGC 
PKN1AGC 
PKN2AGC 
CAMK2DCAMK 
CHEK1CAMK 
DAPK2CAMK 
DAPK3CAMK 
STK17ACAMK 
STK17BCAMK 
PHKG1CAMK 
PHKG2CAMK 
PIM1CAMK 
PIM3CAMK 
PRKD3CAMK 
CHEK2CAMK 
CDK2CMGC 
CDK3CMGC 
CDK9CMGC 
CDC2L5CMGC 
CDKL2CMGC 
CDKL3CMGC 
CDKL5CMGC 
GSK3ACMGC 
ICKCMGC 
AURKCOther 
JAK3TK 
RETTK 
BRAFTKL 

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
AKT1AGC    
AKT2AGC    
AKT3AGC    
GRK4AGC    
GRK7AGC    
PKN1AGC    
PKN2AGC    
PRKACAAGC    
PRKCBAGC    
PRKCBAGC    
PRKCDAGC    
PRKCEAGC    
PRKCHAGC    
PRKCQAGC    
PRKG1AGC    
PRKG2AGC    
PRKXAGC    
ROCK1AGC    
CAMK2DCAMK    
CHEK1CAMK    
CHEK2CAMK    
DAPK2CAMK    
DAPK3CAMK    
PHKG1CAMK    
PHKG2CAMK    
PIM1CAMK    
PIM3CAMK    
PRKD3CAMK    
STK17ACAMK    
CDK2CMGC    
CDK3CMGC    
CDK9CMGC    
GSK3ACMGC    
AURKCOther    
JAK3TK    
RETTK    
BRAFTKL