Kinase profiling results of kinases in KIF 2ZB1A_GK4 (MAPK14, PDB code: 2ZB1, chain A)
Template Kinase: MAPK14
Template inhibitor: biphenyl amide, 4

55 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C
GRK7AGC   
PDPK1AGC   
RPS6KA1AGC   
RPS6KA1CAMK   
RPS6KA2AGC   
RPS6KA2CAMK   
RPS6KA3AGC   
RPS6KA6AGC   
RPS6KA6CAMK   
CHEK1CAMK   
MARK1CAMK   
MARK2CAMK   
MARK3CAMK   
MARK4CAMK   
NUAK1CAMK   
NUAK2CAMK   
SIK1CAMK   
SIK2CAMK   
DAPK1CAMK   
DAPK2CAMK   
DAPK3CAMK   
STK17ACAMK   
STK17BCAMK   
PHKG1CAMK   
PHKG2CAMK   
PRKD1CAMK   
PRKD2CAMK   
PRKD3CAMK   
TSSK1BCAMK   
CDK2CMGC   
CSNK2A2CMGC   
CLK2CMGC   
HIPK2CMGC   
HIPK3CMGC   
PRPF4BCMGC   
GSK3ACMGC   
GSK3BCMGC   
MAPK10CMGC   
MAPK8CMGC   
MAPK9CMGC   
MAPK11CMGC   
MAPK14CMGC   
SLKSTE   
STK10STE   
STK24STE   
ABL1TK   
ABL2TK   
EPHB2TK   
FGFR1TK   
FGFR2TK   
FGRTK   
FYNTK   
SRCTK   
YES1TK   
BLKTK   
HCKTK   
LCKTK   
LYNTK   

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C
GRK7AGC  
PDPK1AGC  
RPS6KA1AGC  
RPS6KA2AGC  
RPS6KA3AGC  
RPS6KA6AGC  
CHEK1CAMK  
DAPK1CAMK  
DAPK2CAMK  
DAPK3CAMK  
MARK1CAMK  
MARK2CAMK  
MARK3CAMK  
MARK4CAMK  
NUAK1CAMK  
NUAK2CAMK  
PHKG1CAMK  
PHKG2CAMK  
PRKD1CAMK  
PRKD2CAMK  
PRKD3CAMK  
SIK2CAMK  
STK17ACAMK  
TSSK1BCAMK  
CDK2CMGC  
CLK2CMGC  
CSNK2A2CMGC  
GSK3ACMGC  
GSK3BCMGC  
HIPK2CMGC  
HIPK3CMGC  
MAPK10CMGC  
MAPK11CMGC  
MAPK14CMGC  
MAPK8CMGC  
MAPK9CMGC  
SLKSTE  
STK10STE  
STK24STE  
ABL1TK  
ABL2TK  
BLKTK  
EPHB2TK  
FGFR1TK  
FGFR2TK  
FGRTK  
FYNTK  
HCKTK  
LCKTK  
LYNTK  
SRCTK  
YES1TK