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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
BMX (
P51813
)
Kinase group
TK
Number of conformation types
0
Number of structural templates
88 (
Total 58 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
55
1BYGA_STU
(CSK)
TK
staurosporine
I
85
72
123
A
1BYGA_STU
(CSK)
TK
staurosporine
I
85
72
123
85
72
123
A
1U59A_STU
(ZAP70)
TK
staurosporine
I
96
80
114
96
80
114
A
3A4OX_STU
(LYN)
TK
staurosporine
I
73
70
88
73
70
88
A
1XBCA_STU
(SYK)
TK
staurosporine
I
71
72
105
71
72
105
A
1YVJA_4ST
(JAK3)
TK
staurosporine
I
96
90
126
96
90
126
A
1QPDA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
2DQ7X_STU
(FYN)
TK
staurosporine
I
91
74
124
91
74
124
A
1QPJA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
2HZ4A_4ST
(ABL1)
TK
staurosporine
I
159
103
156
159
103
156
A
3CKXA_STU
(STK24)
TK
staurosporine
I
176
104
141
176
104
141
A
1SM2A_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1AQ1A_STU
(CDK2)
TK
staurosporine
I
195
76
118
195
76
118
A
1SNUA_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1PKDA_UCN
(CDK2)
TK
UCN 02
I
195
67
118
195
67
118
A
2IVUA_ZD6
(RET)
TK
Vandetanib
I
83
291
121
83
291
121
A
2GQGA_1N1
(ABL1)
TK
Dasatinib
I
74
32
117
74
32
117
A
3K54A_1N1
(BTK)
TK
Dasatinib
I
56
32
103
56
32
103
A
3OCTA_1N1
(BTK)
TK
Dasatinib
I
56
32
103
56
32
103
A
2F4JA_VX6
(ABL1)
TK
VX-680
I
110
109
134
110
109
134
A
2WIHA_P48
(CDK2)
TK
VX_680
I
111
425
105
111
425
105
A
2XYNA_VX6
(ABL2)
TK
VX-680
I
79
101
105
79
101
105
A
3E5AA_VX6
(AURKA)
TK
VX-680
I
57
107
93
57
107
93
A
2X81A_ZZL
(AURKA)
TK
MLN8054
I
22
24
64
22
24
64
A
2IW6A_QQ2
(CDK2)
TK
2iw6
I
112
209
86
112
209
86
A
2H8HA_H8H
(SRC)
TK
Saracatinib
I
91
255
126
91
255
126
A
2J51A_DKI
(SLK)
TK
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2JFLA_DKI
(SLK)
TK
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2R3NA_SCZ
(CDK2)
TK
AC1LZZHM
I
46
175
57
46
175
57
A
1OGUA_ST8
(CDK2)
TK
ST8
I
31
21
34
31
21
34
A
3PJ3A_04L
(BTK)
TK
Imatinib
II
99
113
134
99
113
134
A
2ZYBA_KSL
(LCK)
TK
DB08056
I
36
172
80
36
172
80
A
1OIYA_N41
(CDK2)
TK
N41
I
33
49
34
33
49
34
A
1OPLA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
3B2WA_9NH
(LCK)
TK
MLS000911569
II
30
32
98
30
32
98
A
3GENA_B43
(BTK)
TK
7-Cyclopenty...
I
29
110
67
29
110
67
A
3EJ1A_5BP
(CDK2)
TK
AC1OCFRV
I
46
92
62
46
92
62
A
2FO0A_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
3KMMA_LHL
(LCK)
TK
AZD_1152HQPA
I
29
99
95
29
99
95
A
1QCFA_PP1
(HCK)
TK
PP1
I
31
65
68
31
65
68
A
3GXLA_QIG
(TGFBR1)
TK
DB08450
I
7
34
15
7
34
15
A
2G2HA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
3PJ1A_LHL
(BTK)
TK
AZD_1152HQPA
I
30
99
96
30
99
96
A
1QPEA_PP2
(LCK)
TK
AG 1879
I
29
63
51
29
63
51
A
3HMMA_855
(TGFBR1)
TK
DB07267
I
8
34
22
8
34
22
A
2IW8A_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
2HZIA_JIN
(ABL1)
TK
PD180970
I
90
77
120
90
77
120
A
2IVVA_PP1
(RET)
TK
PP1
I
27
46
63
27
46
63
A
2IW9A_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
3FQSA_585
(SYK)
TK
R-406
I
64
28
102
64
28
102
A
3RI1A_3RH
(FGFR2)
TK
6-o-tolylqui...
I
29
33
72
29
33
72
A
2BHEA_BRY
(CDK2)
TK
BRY
I
51
31
35
51
31
35
A
3IKAA_0UN
(EGFR)
TK
2jkk
I
76
120
108
76
120
108
A
3B8RA_887
(KDR)
TK
3b8r
II
4
32
7
4
32
7
A
1H1SA_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
3PIYA_585
(BTK)
TK
R-406
I
93
17
123
93
17
123
B
30
2ITWA_STU
(EGFR)
TK
staurosporine
I
80
85
106
B
2ITWA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
1OKYA_STU
(PDPK1)
TK
staurosporine
I
179
67
109
179
67
109
B
1WVYA_STU
(DAPK1)
TK
staurosporine
I
83
23
55
83
23
55
B
3BKBA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
2ITQA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
3D7TA_STU
(CSK)
TK
staurosporine
I
70
68
99
70
68
99
B
2ITUA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
3LCSA_STU
(ALK)
TK
staurosporine
I
73
100
109
73
100
109
B
1OKZA_UCN
(PDPK1)
TK
UCN 02
I
179
60
109
179
60
109
B
2ITZA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITOA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITYA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2WTWA_ZZL
(AURKA)
TK
MLN8054
I
35
24
70
35
24
70
B
3H10A_97B
(AURKA)
TK
MLN8054
I
39
88
82
39
88
82
B
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
77
287
111
B
1H07A_MFP
(CDK2)
TK
AC1NAKJQ
I
90
241
80
90
241
80
B
3F5PA_741
(IGF1R)
TK
3-cyanoquino...
I
60
123
81
60
123
81
B
2XB7A_GUI
(ALK)
TK
NVP-TAE684
I
71
66
107
71
66
107
B
3EKNA_GS3
(INSR)
TK
pyrrolo[2,3-...
I
90
215
127
90
215
127
B
2J5FA_DJK
(EGFR)
TK
4-anilinoqui...
I
16
212
45
16
212
45
B
2VX1A_7X8
(EPHB4)
TK
DB07256
I
19
37
15
19
37
15
B
3EFWA_AK8
(AURKA)
TK
3efw
I
100
59
105
100
59
105
B
3COHA_83H
(AURKA)
TK
AKI-001
I
79
88
65
79
88
65
B
2C6IA_DT1
(CDK2)
TK
2c6i
I
27
41
48
27
41
48
B
2C6OA_4SP
(CDK2)
TK
nu6102
I
23
33
27
23
33
27
B
3NRMA_NRM
(AURKA)
TK
CAS404828_08_6
I
32
33
60
32
33
60
B
3P9JA_P9J
(AURKA)
TK
4-[(5-Methyl...
I
32
50
54
32
50
54
B
3LW0A_CCX
(IGF1R)
TK
5-vinyl-3-py...
III
53
30
101
53
30
101
E
3
2HIWA_7MP
(ABL1)
TK
2hiw
II
16
47
53
E
2HIWA_7MP
(ABL1)
TK
2hiw
II
16
47
53
16
47
53
E
2OFVA_242
(LCK)
TK
2ofv
II
28
181
65
28
181
65
E
2OG8A_1N8
(LCK)
TK
1N8
II
35
190
69
35
190
69