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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
CDK3 (
Q00526
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
89 (
Total 38 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
53
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1QPDA_STU
(LCK)
CMGC
staurosporine
I
115
76
126
115
76
126
A
2HY81_1ST
(PAK1)
CMGC
UCN 02
I
58
20
75
58
20
75
A
3HMOA_STU
(TTK)
CMGC
staurosporine
I
27
50
20
27
50
20
A
1BYGA_STU
(CSK)
CMGC
staurosporine
I
85
72
123
85
72
123
A
1QPJA_STU
(LCK)
CMGC
staurosporine
I
115
76
126
115
76
126
A
2HZ4A_4ST
(ABL1)
CMGC
staurosporine
I
159
103
156
159
103
156
A
1NVQA_UCN
(CHEK1)
CMGC
UCN 02
I
179
65
79
179
65
79
A
1SM2A_STU
(ITK)
CMGC
staurosporine
I
99
104
128
99
104
128
A
3A4OX_STU
(LYN)
CMGC
staurosporine
I
73
70
88
73
70
88
A
1NVRA_STU
(CHEK1)
CMGC
staurosporine
I
179
71
79
179
71
79
A
1SNUA_STU
(ITK)
CMGC
staurosporine
I
99
104
128
99
104
128
A
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
121
101
106
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
1YHSA_STU
(PIM1)
CMGC
staurosporine
I
78
64
50
78
64
50
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
2DQ7X_STU
(FYN)
CMGC
staurosporine
I
91
74
124
91
74
124
A
3FMEA_STU
(MAP2K6)
CMGC
staurosporine
I
28
15
20
28
15
20
A
2JFLA_DKI
(SLK)
CMGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2WU6A_DKI
(CLK3)
CMGC
5-AMINO-3-{[...
I
26
9
26
26
9
26
A
2J51A_DKI
(SLK)
CMGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2Z7SA_P01
(RPS6KA1)
CMGC
Lopac0_000938
I
32
214
49
32
214
49
A
3BLRA_CPB
(CDK9)
CMGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
3EQFA_KSA
(MAP2K1)
CMGC
k-252a
I
42
51
57
42
51
57
A
1R0EA_DFN
(GSK3B)
CMGC
HMS3401D14
I
17
17
17
17
17
17
A
3DOGA_NNN
(CDK2)
CMGC
NSC743927
I
50
239
48
50
239
48
A
2JDRA_L20
(AKT2)
CMGC
A-443654
I
44
255
61
44
255
61
A
1Q3WA_ATU
(GSK3B)
CMGC
alsterpaullone
I
24
28
19
24
28
19
A
2BIKB_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
A
1BL7A_SB4
(MAPK14)
CMGC
SB220025
I
22
159
29
22
159
29
A
2ZM4A_KSM
(LCK)
CMGC
BMS-279700
I
25
179
75
25
179
75
A
2BRNA_DF1
(CHEK1)
CMGC
pyrrolopyrim...
I
30
119
42
30
119
42
A
2BILB_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
A
1G5SA_I17
(CDK2)
CMGC
H724
I
43
170
58
43
170
58
A
3BGQA_VX2
(PIM1)
CMGC
triazolopyri...
I
10
25
14
10
25
14
A
2BROA_DF2
(CHEK1)
CMGC
pyrrolopyrim...
I
29
109
40
29
109
40
A
2I0EA_PDS
(PRKCB)
CMGC
bisindolylma...
I
41
141
45
41
141
45
A
3SD0A_TSK
(GSK3B)
CMGC
3-(5-Fluoro-...
I
9
38
17
9
38
17
A
2JAVA_5Z5
(NEK2)
CMGC
pyrrollylact...
I
25
40
24
25
40
24
A
1OUKA_084
(MAPK14)
CMGC
1ouk
I
24
139
46
24
139
46
A
3OT3A_22K
(CHEK1)
CMGC
INCB18424
I
13
30
13
13
30
13
A
3DDPA_RC8
(CDK2)
CMGC
Roscovitine
I
42
133
57
42
133
57
A
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
62
139
51
A
2VTQA_LZA
(CDK2)
CMGC
pyrazole dia...
I
36
25
31
36
25
31
A
1UV5A_BRW
(GSK3B)
CMGC
6-bromoindir...
I
27
37
28
27
37
28
A
3IW4A_LW4
(PRKCA)
CMGC
Sotrastaurin
I
52
119
49
52
119
49
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
A
2BHEA_BRY
(CDK2)
CMGC
BRY
I
51
31
35
51
31
35
A
2VU3A_LZE
(CDK2)
CMGC
AT7519
I
35
22
29
35
22
29
A
3LQ5A_SLQ
(CDK9)
CMGC
Roscovitine
I
25
130
37
25
130
37
A
3KVWA_IRB
(DYRK2)
CMGC
CI_1040
I
15
36
12
15
36
12
A
1XWSA_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
B
36
3BKBA_STU
(FES)
CMGC
staurosporine
I
131
107
138
B
3BKBA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
1WVYA_STU
(DAPK1)
CMGC
staurosporine
I
83
23
55
83
23
55
B
3CBLA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
3CD3A_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
2W4OA_DKI
(CAMK4)
CMGC
5-AMINO-3-{[...
I
15
9
22
15
9
22
B
3AMAA_SKE
(PRKACA)
CMGC
JNJ-7706621
I
46
26
35
46
26
35
B
2F57B_23D
(PAK7)
CMGC
CGP74514A
I
11
77
24
11
77
24
B
3EFWA_AK8
(AURKA)
CMGC
3efw
I
100
59
105
100
59
105
B
2F2CB_AP9
(CDK6)
CMGC
MLS000911551
I
24
147
39
24
147
39
B
2A0CX_CK9
(CDK2)
CMGC
purine deriv...
I
45
226
50
45
226
50
B
3NS9A_NS9
(CDK2)
CMGC
pyrazolo[1,5...
I
44
196
47
44
196
47
B
2A4LA_RRC
(CDK2)
CMGC
roscovitine
I
50
240
50
50
240
50
B
3PJ8A_404
(CDK2)
CMGC
imidazo[2,1-...
I
47
223
49
47
223
49
B
1CKPA_PVB
(CDK2)
CMGC
Purvalanol B
I
35
76
36
35
76
36
B
3DDQA_RRC
(CDK2)
CMGC
roscovitine
I
50
240
50
50
240
50
B
3NYNA_SGV
(GRK6)
CMGC
SMR000127424
I
54
7
47
54
7
47
B
1UNLA_RRC
(CDK5)
CMGC
roscovitine
I
45
237
47
45
237
47
B
1W0XC_OLO
(CDK2)
CMGC
olomoucine
I
43
195
47
43
195
47
B
2B54A_D05
(CDK2)
CMGC
D05
I
11
33
14
11
33
14
B
1ZRZA_BI1
(PRKCI)
CMGC
bisindolylma...
I
52
150
47
52
150
47
B
2FVDA_LIA
(CDK2)
CMGC
[4-Amino-2-[...
I
39
16
29
39
16
29
B
3L9MA_L9M
(PRKACA)
CMGC
VX_680
I
37
65
42
37
65
42
B
1PF8A_SU9
(CDK2)
CMGC
SU 9516
I
25
19
33
25
19
33
B
3COHA_83H
(AURKA)
CMGC
AKI-001
I
79
88
65
79
88
65
B
3PY0A_SU9
(CDK2)
CMGC
SU 9516
I
25
19
33
25
19
33
B
1UU7A_BI2
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
3PY1A_SU9
(CDK2)
CMGC
SU 9516
I
25
19
33
25
19
33
B
1UU8A_BI1
(PDPK1)
CMGC
bisindolylma...
I
83
189
65
83
189
65
B
1PMNA_984
(MAPK10)
CMGC
1pmn
I
10
124
20
10
124
20
B
1UU9A_BI3
(PDPK1)
CMGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1PMQA_880
(MAPK10)
CMGC
1pmq
I
12
105
20
12
105
20
B
1UVRA_BI8
(PDPK1)
CMGC
Ro 31-7549
I
82
181
65
82
181
65
B
3ORZA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65