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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
CDK8 (
P49336
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
23 (
Total 29 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
9
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
2HY81_1ST
(PAK1)
CMGC
UCN 02
I
58
20
75
58
20
75
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
3BLRA_CPB
(CDK9)
CMGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
3HA8A_5JZ
(MAPK14)
CMGC
DEL-B, 14b
I
59
89
62
59
89
62
A
3I4BA_Z48
(GSK3B)
CMGC
Z48
I
18
77
34
18
77
34
A
3I5ZA_Z48
(MAPK1)
CMGC
Z48
I
12
64
26
12
64
26
B
14
3EFWA_AK8
(AURKA)
CMGC
3efw
I
100
59
105
B
3EFWA_AK8
(AURKA)
CMGC
3efw
I
100
59
105
100
59
105
B
1WVYA_STU
(DAPK1)
CMGC
staurosporine
I
83
23
55
83
23
55
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
2C6EA_HPM
(AURKA)
CMGC
HPM
I
44
237
90
44
237
90
B
2R3FA_SC8
(CDK2)
CMGC
2c68
I
22
62
43
22
62
43
B
2R3GA_SC9
(CDK2)
CMGC
2r3j
I
30
137
50
30
137
50
B
2R3IA_SCF
(CDK2)
CMGC
2c68
I
23
89
43
23
89
43
B
2R3JA_SCJ
(CDK2)
CMGC
2r3j
I
27
99
49
27
99
49
B
2R3KA_SCQ
(CDK2)
CMGC
2r3j
I
28
95
49
28
95
49
B
2R3LA_SCW
(CDK2)
CMGC
2r3j
I
19
63
41
19
63
41
B
2C68A_CT6
(CDK2)
CMGC
2c68
I
23
73
43
23
73
43
B
2R3RA_6SC
(CDK2)
CMGC
2r3j
I
13
55
30
13
55
30
B
2C69A_CT8
(CDK2)
CMGC
CT8
I
22
62
38
22
62
38