BioXGEM.
KIDFamMap
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Example1
Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
CIT (
O14578
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
7 (
Total 71 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
4
2VD5A_BI8
(DMPK)
AGC
Ro 31-7549
I
19
49
12
A
2VD5A_BI8
(DMPK)
AGC
Ro 31-7549
I
19
49
12
19
49
12
A
1XJDA_STU
(PRKCQ)
AGC
staurosporine
I
121
101
106
121
101
106
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
B
3
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
B
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
52
150
47
B
3NYNA_SGV
(GRK6)
AGC
SMR000127424
I
54
7
47
54
7
47
B
3L9MA_L9M
(PRKACA)
AGC
VX_680
I
37
65
42
37
65
42