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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
DYRK1B (
Q9Y463
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
53 (
Total 91 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
30
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
121
101
106
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
2JAMA_J60
(CAMK1G)
CMGC
SU11652
I
50
65
32
50
65
32
A
2XIKA_J60
(STK25)
CMGC
SU11652
I
59
49
65
59
49
65
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
A
2X7GA_PVB
(SRPK2)
CMGC
Purvalanol B
I
3
6
0
3
6
0
A
2J7TA_274
(STK10)
CMGC
SU11274
I
66
20
77
66
20
77
A
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
62
139
51
A
3DOGA_NNN
(CDK2)
CMGC
NSC743927
I
50
239
48
50
239
48
A
3IW4A_LW4
(PRKCA)
CMGC
Sotrastaurin
I
52
119
49
52
119
49
A
1R78A_FMD
(CDK2)
CMGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
3DDPA_RC8
(CDK2)
CMGC
Roscovitine
I
42
133
57
42
133
57
A
3BLRA_CPB
(CDK9)
CMGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
3LQ5A_SLQ
(CDK9)
CMGC
Roscovitine
I
25
130
37
25
130
37
A
2XM8A_B4W
(CHEK2)
CMGC
PI_103
I
12
54
18
12
54
18
A
3ANQA_EHB
(DYRK1A)
CMGC
TG003
I
7
3
2
7
3
2
A
2WU6A_DKI
(CLK3)
CMGC
5-AMINO-3-{[...
I
26
9
26
26
9
26
A
3HA8A_5JZ
(MAPK14)
CMGC
DEL-B, 14b
I
59
89
62
59
89
62
A
1R0EA_DFN
(GSK3B)
CMGC
HMS3401D14
I
17
17
17
17
17
17
A
2VTQA_LZA
(CDK2)
CMGC
pyrazole dia...
I
36
25
31
36
25
31
A
3EIDA_PO5
(CDK2)
CMGC
AC1O6YZF
I
63
211
77
63
211
77
A
2VU3A_LZE
(CDK2)
CMGC
AT7519
I
35
22
29
35
22
29
A
3L8XA_N4D
(MAPK14)
CMGC
3cg2
I
91
104
65
91
104
65
A
2JEDA_LG8
(PRKCQ)
CMGC
5-Arylidene-...
I
67
19
87
67
19
87
A
2O0UA_C0M
(MAPK10)
CMGC
ZINC00799686
I
21
8
23
21
8
23
A
2J51A_DKI
(SLK)
CMGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2JFLA_DKI
(SLK)
CMGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
B
23
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
2PE2A_464
(PDPK1)
CMGC
Indolinone b...
I
134
156
104
134
156
104
B
2A0CX_CK9
(CDK2)
CMGC
purine deriv...
I
45
226
50
45
226
50
B
3NS9A_NS9
(CDK2)
CMGC
pyrazolo[1,5...
I
44
196
47
44
196
47
B
3OTUA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
2A4LA_RRC
(CDK2)
CMGC
roscovitine
I
50
240
50
50
240
50
B
3PJ8A_404
(CDK2)
CMGC
imidazo[2,1-...
I
47
223
49
47
223
49
B
1UU7A_BI2
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
2F2CB_AP9
(CDK6)
CMGC
MLS000911551
I
24
147
39
24
147
39
B
1UU8A_BI1
(PDPK1)
CMGC
bisindolylma...
I
83
189
65
83
189
65
B
1UU9A_BI3
(PDPK1)
CMGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
CMGC
Ro 31-7549
I
82
181
65
82
181
65
B
1CKPA_PVB
(CDK2)
CMGC
Purvalanol B
I
35
76
36
35
76
36
B
3DDQA_RRC
(CDK2)
CMGC
roscovitine
I
50
240
50
50
240
50
B
1UNLA_RRC
(CDK5)
CMGC
roscovitine
I
45
237
47
45
237
47
B
1W0XC_OLO
(CDK2)
CMGC
olomoucine
I
43
195
47
43
195
47
B
3ORZA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU3A_LY4
(PDPK1)
CMGC
Ruboxistaurin
I
71
117
57
71
117
57
B
1OIRA_HDY
(CDK2)
CMGC
AC1O6YZF
I
51
203
64
51
203
64
B
3NAYA_MP6
(PDPK1)
CMGC
ZINC13474643
I
20
81
37
20
81
37
B
2FVDA_LIA
(CDK2)
CMGC
[4-Amino-2-[...
I
39
16
29
39
16
29
B
2R3OA_2SC
(CDK2)
CMGC
4-(Benzylami...
I
18
36
43
18
36
43