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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
PIM3 (
Q86V86
)
Kinase group
CAMK
Number of conformation types
0
Number of structural templates
55 (
Total 77 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
39
1AQ1A_STU
(CDK2)
CAMK
staurosporine
I
195
76
118
A
1AQ1A_STU
(CDK2)
CAMK
staurosporine
I
195
76
118
195
76
118
A
1XJDA_STU
(PRKCQ)
CAMK
staurosporine
I
121
101
106
121
101
106
A
1NVRA_STU
(CHEK1)
CAMK
staurosporine
I
179
71
79
179
71
79
A
1YHSA_STU
(PIM1)
CAMK
staurosporine
I
78
64
50
78
64
50
A
1NXKA_STU
(MAPKAPK2)
CAMK
staurosporine
I
110
67
51
110
67
51
A
3HMOA_STU
(TTK)
CAMK
staurosporine
I
27
50
20
27
50
20
A
1Q3DA_STU
(GSK3B)
CAMK
staurosporine
I
115
71
61
115
71
61
A
1NVQA_UCN
(CHEK1)
CAMK
UCN 02
I
179
65
79
179
65
79
A
1PKDA_UCN
(CDK2)
CAMK
UCN 02
I
195
67
118
195
67
118
A
3JPVA_1DR
(PIM1)
CAMK
1DR
I
5
11
2
5
11
2
A
2BILB_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
2I0EA_PDS
(PRKCB)
CAMK
bisindolylma...
I
41
141
45
41
141
45
A
2OW3A_BIM
(GSK3B)
CAMK
LY_333531
I
62
139
51
62
139
51
A
3IW4A_LW4
(PRKCA)
CAMK
Sotrastaurin
I
52
119
49
52
119
49
A
1XWSA_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
2BIKB_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
2J2IB_LY4
(PIM1)
CAMK
Ruboxistaurin
I
35
89
36
35
89
36
A
2HY81_1ST
(PAK1)
CAMK
UCN 02
I
58
20
75
58
20
75
A
3M2WA_L8I
(MAPKAPK2)
CAMK
Sunitinib
I
84
90
47
84
90
47
A
3BGZA_VX3
(PIM1)
CAMK
2,3-diphenyl...
I
9
14
8
9
14
8
A
2VTTA_LZD
(CDK2)
CAMK
pyrazole dia...
I
158
42
111
158
42
111
A
1R78A_FMD
(CDK2)
CAMK
4-alkynyl ox...
I
127
24
97
127
24
97
A
3CY3A_JN5
(PIM1)
CAMK
JN5
I
8
10
10
8
10
10
A
2ZV2A_609
(CAMKK2)
CAMK
STO-609
I
10
11
10
10
11
10
A
2V7OA_DRN
(CAMK2G)
CAMK
bisindolylma...
I
23
51
16
23
51
16
A
2Z7SA_P01
(RPS6KA1)
CAMK
Lopac0_000938
I
32
214
49
32
214
49
A
1YI3A_LY2
(PIM1)
CAMK
LY294002
I
3
2
2
3
2
2
A
3BGQA_VX2
(PIM1)
CAMK
triazolopyri...
I
10
25
14
10
25
14
A
2UZEA_C95
(CDK2)
CAMK
STK004775
I
4
9
6
4
9
6
A
3OT3A_22K
(CHEK1)
CAMK
INCB18424
I
13
30
13
13
30
13
A
2JDRA_L20
(AKT2)
CAMK
A-443654
I
44
255
61
44
255
61
A
2J90A_IZA
(DAPK3)
CAMK
Pyridone 6
I
40
50
42
40
50
42
A
2BHEA_BRY
(CDK2)
CAMK
BRY
I
51
31
35
51
31
35
A
3JYAA_LWG
(PIM1)
CAMK
Kinome_3259
I
4
5
1
4
5
1
A
1Q3WA_ATU
(GSK3B)
CAMK
alsterpaullone
I
24
28
19
24
28
19
A
1NVSA_UCM
(CHEK1)
CAMK
SB218078
I
97
6
53
97
6
53
A
2I40A_BLZ
(CDK2)
CAMK
2i40
I
34
95
16
34
95
16
A
3D0EA_G93
(AKT2)
CAMK
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
1G5SA_I17
(CDK2)
CAMK
H724
I
43
170
58
43
170
58
B
16
1WVYA_STU
(DAPK1)
CAMK
staurosporine
I
83
23
55
B
1WVYA_STU
(DAPK1)
CAMK
staurosporine
I
83
23
55
83
23
55
B
1OKYA_STU
(PDPK1)
CAMK
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CAMK
UCN 02
I
179
60
109
179
60
109
B
1UU9A_BI3
(PDPK1)
CAMK
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
CAMK
Ro 31-7549
I
82
181
65
82
181
65
B
1UU7A_BI2
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
CAMK
bisindolylma...
I
83
189
65
83
189
65
B
3ORZA_BI4
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
1UU3A_LY4
(PDPK1)
CAMK
Ruboxistaurin
I
71
117
57
71
117
57
B
1H00A_FAP
(CDK2)
CAMK
AC1NAE4F
I
50
94
75
50
94
75
B
2PE2A_464
(PDPK1)
CAMK
Indolinone b...
I
134
156
104
134
156
104
B
3NYNA_SGV
(GRK6)
CAMK
SMR000127424
I
54
7
47
54
7
47
B
2W1FA_L0F
(AURKA)
CAMK
DB08066
I
17
40
35
17
40
35
B
3COHA_83H
(AURKA)
CAMK
AKI-001
I
79
88
65
79
88
65
B
2W1HA_L0H
(CDK2)
CAMK
DB08066
I
20
43
42
20
43
42