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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
6 PRKACB related diseases
hsa05020
Prion diseases
hsa05030
Cocaine addiction
hsa05110
Vibrio cholerae infection
hsa05146
Amoebiasis
hsa05169
Epstein-Barr virus infection
hsa05414
Dilated cardiomyopathy
Summary of query kinase
Query kinase
PRKACB (
P22694
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
26 (
Total 23 inhibitors
)
Number of PRKACB related diseases
6 (
hsa05020
hsa05030
hsa05110
hsa05146
hsa05169
hsa05414
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
9
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
2HZ4A_4ST
(ABL1)
AGC
staurosporine
I
159
103
156
159
103
156
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
1BL6A_SB6
(MAPK14)
AGC
sb216995
I
46
110
50
46
110
50
A
1OZ1A_FPH
(MAPK14)
AGC
4-Azaindole 6
I
18
27
28
18
27
28
A
3FKOA_FKO
(MAPK14)
AGC
L-779450
I
17
7
27
17
7
27
A
3HA8A_5JZ
(MAPK14)
AGC
DEL-B, 14b
I
59
89
62
59
89
62
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
B
17
3CD3A_STU
(FES)
AGC
staurosporine
I
131
107
138
B
3CD3A_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
1WVYA_STU
(DAPK1)
AGC
staurosporine
I
83
23
55
83
23
55
B
3BKBA_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
52
150
47
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
3EFWA_AK8
(AURKA)
AGC
3efw
I
100
59
105
100
59
105
B
3NYNA_SGV
(GRK6)
AGC
SMR000127424
I
54
7
47
54
7
47
B
3L9MA_L9M
(PRKACA)
AGC
VX_680
I
37
65
42
37
65
42