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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
STK17A (
Q9UEE5
)
Kinase group
CAMK
Number of conformation types
0
Number of structural templates
80 (
Total 73 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
56
1PKDA_UCN
(CDK2)
CAMK
UCN 02
I
195
67
118
A
1PKDA_UCN
(CDK2)
CAMK
UCN 02
I
195
67
118
195
67
118
A
2HW7A_STU
(MKNK2)
CAMK
staurosporine
I
28
55
16
28
55
16
A
1QPDA_STU
(LCK)
CAMK
staurosporine
I
115
76
126
115
76
126
A
2JAMA_J60
(CAMK1G)
CAMK
SU11652
I
50
65
32
50
65
32
A
1AQ1A_STU
(CDK2)
CAMK
staurosporine
I
195
76
118
195
76
118
A
1QPJA_STU
(LCK)
CAMK
staurosporine
I
115
76
126
115
76
126
A
3A4OX_STU
(LYN)
CAMK
staurosporine
I
73
70
88
73
70
88
A
2XIKA_J60
(STK25)
CAMK
SU11652
I
59
49
65
59
49
65
A
1NVQA_UCN
(CHEK1)
CAMK
UCN 02
I
179
65
79
179
65
79
A
1U59A_STU
(ZAP70)
CAMK
staurosporine
I
96
80
114
96
80
114
A
3CKXA_STU
(STK24)
CAMK
staurosporine
I
176
104
141
176
104
141
A
1NVRA_STU
(CHEK1)
CAMK
staurosporine
I
179
71
79
179
71
79
A
1XBCA_STU
(SYK)
CAMK
staurosporine
I
71
72
105
71
72
105
A
3FMEA_STU
(MAP2K6)
CAMK
staurosporine
I
28
15
20
28
15
20
A
1NXKA_STU
(MAPKAPK2)
CAMK
staurosporine
I
110
67
51
110
67
51
A
1XJDA_STU
(PRKCQ)
CAMK
staurosporine
I
121
101
106
121
101
106
A
1YHSA_STU
(PIM1)
CAMK
staurosporine
I
78
64
50
78
64
50
A
1YVJA_4ST
(JAK3)
CAMK
staurosporine
I
96
90
126
96
90
126
A
2J7TA_274
(STK10)
CAMK
SU11274
I
66
20
77
66
20
77
A
2HY81_1ST
(PAK1)
CAMK
UCN 02
I
58
20
75
58
20
75
A
2VTTA_LZD
(CDK2)
CAMK
pyrazole dia...
I
158
42
111
158
42
111
A
3M2WA_L8I
(MAPKAPK2)
CAMK
Sunitinib
I
84
90
47
84
90
47
A
1XBBA_STI
(SYK)
CAMK
Imatinib
I
31
170
75
31
170
75
A
1R78A_FMD
(CDK2)
CAMK
4-alkynyl ox...
I
127
24
97
127
24
97
A
3EQFA_KSA
(MAP2K1)
CAMK
k-252a
I
42
51
57
42
51
57
A
2J51A_DKI
(SLK)
CAMK
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2JFLA_DKI
(SLK)
CAMK
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2X81A_ZZL
(AURKA)
CAMK
MLN8054
I
22
24
64
22
24
64
A
3HA8A_5JZ
(MAPK14)
CAMK
DEL-B, 14b
I
59
89
62
59
89
62
A
2JEDA_LG8
(PRKCQ)
CAMK
5-Arylidene-...
I
67
19
87
67
19
87
A
3EIDA_PO5
(CDK2)
CAMK
AC1O6YZF
I
63
211
77
63
211
77
A
3L8XA_N4D
(MAPK14)
CAMK
3cg2
I
91
104
65
91
104
65
A
2I0EA_PDS
(PRKCB)
CAMK
bisindolylma...
I
41
141
45
41
141
45
A
1NVSA_UCM
(CHEK1)
CAMK
SB218078
I
97
6
53
97
6
53
A
1OI9A_N20
(CDK2)
CAMK
NU-6086
I
52
80
61
52
80
61
A
2VD5A_BI8
(DMPK)
CAMK
Ro 31-7549
I
19
49
12
19
49
12
A
3A2CA_PDY
(MAPKAPK2)
CAMK
6-(4-methoxy...
I
32
39
21
32
39
21
A
3IW4A_LW4
(PRKCA)
CAMK
Sotrastaurin
I
52
119
49
52
119
49
A
1BL6A_SB6
(MAPK14)
CAMK
sb216995
I
46
110
50
46
110
50
A
2BHEA_BRY
(CDK2)
CAMK
BRY
I
51
31
35
51
31
35
A
1ZZLA_TZY
(MAPK14)
CAMK
CP-808844
I
36
84
44
36
84
44
A
3BLRA_CPB
(CDK9)
CAMK
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
2ZB1A_GK4
(MAPK14)
CAMK
biphenyl ami...
II
55
57
54
55
57
54
A
1XWSA_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
3FQSA_585
(SYK)
CAMK
R-406
I
64
28
102
64
28
102
A
2JDRA_L20
(AKT2)
CAMK
A-443654
I
44
255
61
44
255
61
A
2J90A_IZA
(DAPK3)
CAMK
Pyridone 6
I
40
50
42
40
50
42
A
3E92A_G6A
(MAPK14)
CAMK
3e92
I
56
59
55
56
59
55
A
2BIKB_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
2WIHA_P48
(CDK2)
CAMK
VX_680
I
111
425
105
111
425
105
A
3ITZA_P66
(MAPK14)
CAMK
P66
II
15
102
25
15
102
25
A
3LXLA_IZA
(JAK3)
CAMK
Pyridone 6
I
30
11
63
30
11
63
A
2HOGA_710
(CHEK1)
CAMK
3-(Indol-2-y...
I
33
66
51
33
66
51
A
3IPHA_G11
(MAPK14)
CAMK
HMS3303K05
I
57
108
55
57
108
55
A
2BILB_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
3E5AA_VX6
(AURKA)
CAMK
VX-680
I
57
107
93
57
107
93
B
24
1OKYA_STU
(PDPK1)
CAMK
staurosporine
I
179
67
109
B
1OKYA_STU
(PDPK1)
CAMK
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CAMK
UCN 02
I
179
60
109
179
60
109
B
2PE2A_464
(PDPK1)
CAMK
Indolinone b...
I
134
156
104
134
156
104
B
2XCKA_MH4
(PDPK1)
CAMK
MH4
I
46
431
75
46
431
75
B
1H00A_FAP
(CDK2)
CAMK
AC1NAE4F
I
50
94
75
50
94
75
B
2WTWA_ZZL
(AURKA)
CAMK
MLN8054
I
35
24
70
35
24
70
B
3H10A_97B
(AURKA)
CAMK
MLN8054
I
39
88
82
39
88
82
B
3NYNA_SGV
(GRK6)
CAMK
SMR000127424
I
54
7
47
54
7
47
B
1PF8A_SU9
(CDK2)
CAMK
SU 9516
I
25
19
33
25
19
33
B
3PY0A_SU9
(CDK2)
CAMK
SU 9516
I
25
19
33
25
19
33
B
1UU7A_BI2
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
2PE0A_39Z
(PDPK1)
CAMK
2pe0
I
20
2
27
20
2
27
B
3PY1A_SU9
(CDK2)
CAMK
SU 9516
I
25
19
33
25
19
33
B
1UU8A_BI1
(PDPK1)
CAMK
bisindolylma...
I
83
189
65
83
189
65
B
3H9OA_9BD
(PDPK1)
CAMK
Benzo[c][2,7...
I
45
68
71
45
68
71
B
1UU9A_BI3
(PDPK1)
CAMK
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
3ORZA_BI4
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
3COHA_83H
(AURKA)
CAMK
AKI-001
I
79
88
65
79
88
65
B
1UVRA_BI8
(PDPK1)
CAMK
Ro 31-7549
I
82
181
65
82
181
65
B
3OTUA_BI4
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
2B7AA_IZA
(JAK2)
CAMK
Pyridone 6
I
34
12
65
34
12
65
B
3MTLA_FEF
(PCTK1)
CAMK
indirubin de...
I
16
3
23
16
3
23
B
1OIRA_HDY
(CDK2)
CAMK
AC1O6YZF
I
51
203
64
51
203
64
B
2BMCA_MPY
(AURKA)
CAMK
PHA-680632
I
107
108
107
107
108
107