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Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
LZE
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
CDK2 (PDB code: 2VU3)
[PDB]
[PDBsum]
Inhibitor
AT7519 (HET code: LZE)
[PDB]
Summary of KIF 2VU3A_LZE
(CDK2, PDB code:
2VU3
, chain A)
Number of family interactions
59
Number of family kinase
35 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
22 (1 are CDC2L6 inhibitors)
Involved diseases
29 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
CDC2L6 and 1 inhibitors