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Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
L20
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
AKT2 (PDB code: 2JDR)
[PDB]
[PDBsum]
Inhibitor
A-443654 (HET code: L20)
[PDB]
Summary of KIF 2JDRA_L20
(AKT2, PDB code:
2JDR
, chain A)
Number of family interactions
349
Number of family kinase
44 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
255 (1 are CDKL2 inhibitors)
Involved diseases
61 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
CDKL2 and 1 inhibitors