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KIDFamMap
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
KSA
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
MAP2K1 (PDB code: 3EQF)
[PDB]
[PDBsum]
Inhibitor
k-252a (HET code: KSA)
[PDB]
Summary of KIF 3EQFA_KSA
(MAP2K1, PDB code:
3EQF
, chain A)
Number of family interactions
194
Number of family kinase
42 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
51 (2 are CDKL2 inhibitors)
Involved diseases
57 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
CDKL2 and 2 inhibitors