BioXGEM.
KIDFamMap
Home
Example1
Example2
Statistics
Document
Contact US
Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
VX6
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
ABL1 (PDB code: 2F4J)
[PDB]
[PDBsum]
Inhibitor
VX-680 (HET code: VX6)
[PDB]
Summary of KIF 2F4JA_VX6
(ABL1, PDB code:
2F4J
, chain A)
Number of family interactions
546
Number of family kinase
110 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
109 (1 are CDKL5 inhibitors)
Involved diseases
134 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
CDKL5 and 1 inhibitors