Protein Surface  Ribbon
Inhibitor GS3
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase INSR (PDB code: 3EKN) [PDB] [PDBsum]
Inhibitor pyrrolo[2,3-d]pyrimidine deriv., 1 (HET code: GS3) [PDB]
 
Summary of KIF 3EKNA_GS3 (INSR, PDB code: 3EKN, chain A)
Number of family interactions 403
Number of family kinase 90 (sequence conservation) (profiling results)
Number of family inhibitors 215 (1 are DDR2 inhibitors)
Involved diseases 127 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  DDR2 and 1 inhibitors