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Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
PP2
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
LCK (PDB code: 1QPE)
[PDB]
[PDBsum]
Inhibitor
AG 1879 (HET code: PP2)
[PDB]
Summary of KIF 1QPEA_PP2
(LCK, PDB code:
1QPE
, chain A)
Number of family interactions
99
Number of family kinase
29 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
63 (1 are EPHB2 inhibitors)
Involved diseases
51 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
EPHB2 and 1 inhibitors