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KIDFamMap
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
LW4
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
PRKCA (PDB code: 3IW4)
[PDB]
[PDBsum]
Inhibitor
Sotrastaurin (HET code: LW4)
[PDB]
Summary of KIF 3IW4A_LW4
(PRKCA, PDB code:
3IW4
, chain A)
Number of family interactions
479
Number of family kinase
52 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
119 (3 are GRK7 inhibitors)
Involved diseases
49 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
GRK7 and 3 inhibitors