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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
BI8
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
PDPK1 (PDB code: 1UVR)
[PDB]
[PDBsum]
Inhibitor
Ro 31-7549 (HET code: BI8)
[PDB]
Summary of KIF 1UVRA_BI8
(PDPK1, PDB code:
1UVR
, chain A)
Number of family interactions
628
Number of family kinase
82 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
181 (7 are RPS6KA6 inhibitors)
Involved diseases
65 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
RPS6KA6 and 7 inhibitors