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Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
2 GRK1 related diseases
H00787
Congenital stationary night blindness (CSNB)
613411
Oguchi disease-2
Summary of query kinase
Query kinase
GRK1 (
Q15835
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
42 (
Total 24 inhibitors
)
Number of GRK1 related diseases
2 (
H00787
613411
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
25
3FMEA_STU
(MAP2K6)
AGC
staurosporine
I
28
15
20
A
3FMEA_STU
(MAP2K6)
AGC
staurosporine
I
28
15
20
28
15
20
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
1Q3DA_STU
(GSK3B)
AGC
staurosporine
I
115
71
61
115
71
61
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
2XIKA_J60
(STK25)
AGC
SU11652
I
59
49
65
59
49
65
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1XJDA_STU
(PRKCQ)
AGC
staurosporine
I
121
101
106
121
101
106
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
1YVJA_4ST
(JAK3)
AGC
staurosporine
I
96
90
126
96
90
126
A
1NXKA_STU
(MAPKAPK2)
AGC
staurosporine
I
110
67
51
110
67
51
A
3CKXA_STU
(STK24)
AGC
staurosporine
I
176
104
141
176
104
141
A
2J7TA_274
(STK10)
AGC
SU11274
I
66
20
77
66
20
77
A
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
41
141
45
A
3EQFA_KSA
(MAP2K1)
AGC
k-252a
I
42
51
57
42
51
57
A
2OW3A_BIM
(GSK3B)
AGC
LY_333531
I
62
139
51
62
139
51
A
2VTTA_LZD
(CDK2)
AGC
pyrazole dia...
I
158
42
111
158
42
111
A
3IW4A_LW4
(PRKCA)
AGC
Sotrastaurin
I
52
119
49
52
119
49
A
3M2WA_L8I
(MAPKAPK2)
AGC
Sunitinib
I
84
90
47
84
90
47
A
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
17
127
29
A
3GU8A_3GU
(DAPK1)
AGC
Vidarabine
I
14
17
24
14
17
24
A
1R78A_FMD
(CDK2)
AGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
2JEDA_LG8
(PRKCQ)
AGC
5-Arylidene-...
I
67
19
87
67
19
87
A
2O0UA_C0M
(MAPK10)
AGC
ZINC00799686
I
21
8
23
21
8
23
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
2V7OA_DRN
(CAMK2G)
AGC
bisindolylma...
I
23
51
16
23
51
16
B
17
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
1WVYA_STU
(DAPK1)
AGC
staurosporine
I
83
23
55
83
23
55
B
3NYNA_SGV
(GRK6)
AGC
SMR000127424
I
54
7
47
54
7
47
B
2PE2A_464
(PDPK1)
AGC
Indolinone b...
I
134
156
104
134
156
104
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
52
150
47
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
2EVAA_ADN
(MAP3K7)
AGC
Vidarabine
I
6
7
30
6
7
30
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
3KRXA_BA1
(ADRBK1)
AGC
balanol
I
14
106
29
14
106
29
B
2BMCA_MPY
(AURKA)
AGC
PHA-680632
I
107
108
107
107
108
107
B
1MUOA_ADN
(AURKA)
AGC
Vidarabine
I
11
12
32
11
12
32