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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
CDKL2 (
Q92772
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
64 (
Total 26 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
44
2JAMA_J60
(CAMK1G)
CMGC
SU11652
I
50
65
32
A
2JAMA_J60
(CAMK1G)
CMGC
SU11652
I
50
65
32
50
65
32
A
2XIKA_J60
(STK25)
CMGC
SU11652
I
59
49
65
59
49
65
A
2J7TA_274
(STK10)
CMGC
SU11274
I
66
20
77
66
20
77
A
2JAVA_5Z5
(NEK2)
CMGC
pyrrollylact...
I
25
40
24
25
40
24
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
A
2OFUA_1N9
(LCK)
CMGC
2-aminopyrim...
I
55
215
101
55
215
101
A
3EQFA_KSA
(MAP2K1)
CMGC
k-252a
I
42
51
57
42
51
57
A
1AGWA_SU2
(FGFR1)
CMGC
SU 4984
I
77
81
111
77
81
111
A
3IW4A_LW4
(PRKCA)
CMGC
Sotrastaurin
I
52
119
49
52
119
49
A
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
121
101
106
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
1YHSA_STU
(PIM1)
CMGC
staurosporine
I
78
64
50
78
64
50
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
2JEDA_LG8
(PRKCQ)
CMGC
5-Arylidene-...
I
67
19
87
67
19
87
A
1XWSA_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
1YVJA_4ST
(JAK3)
CMGC
staurosporine
I
96
90
126
96
90
126
A
3FMEA_STU
(MAP2K6)
CMGC
staurosporine
I
28
15
20
28
15
20
A
2VTQA_LZA
(CDK2)
CMGC
pyrazole dia...
I
36
25
31
36
25
31
A
2O0UA_C0M
(MAPK10)
CMGC
ZINC00799686
I
21
8
23
21
8
23
A
3PIYA_585
(BTK)
CMGC
R-406
I
93
17
123
93
17
123
A
1QPDA_STU
(LCK)
CMGC
staurosporine
I
115
76
126
115
76
126
A
2HY81_1ST
(PAK1)
CMGC
UCN 02
I
58
20
75
58
20
75
A
1R78A_FMD
(CDK2)
CMGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
2VU3A_LZE
(CDK2)
CMGC
AT7519
I
35
22
29
35
22
29
A
3L8XA_N4D
(MAPK14)
CMGC
3cg2
I
91
104
65
91
104
65
A
2BIKB_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1QPJA_STU
(LCK)
CMGC
staurosporine
I
115
76
126
115
76
126
A
2HZ4A_4ST
(ABL1)
CMGC
staurosporine
I
159
103
156
159
103
156
A
2F4JA_VX6
(ABL1)
CMGC
VX-680
I
110
109
134
110
109
134
A
3PJ3A_04L
(BTK)
CMGC
Imatinib
II
99
113
134
99
113
134
A
2BILB_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
A
1NVQA_UCN
(CHEK1)
CMGC
UCN 02
I
179
65
79
179
65
79
A
1SM2A_STU
(ITK)
CMGC
staurosporine
I
99
104
128
99
104
128
A
3A4OX_STU
(LYN)
CMGC
staurosporine
I
73
70
88
73
70
88
A
2WIHA_P48
(CDK2)
CMGC
VX_680
I
111
425
105
111
425
105
A
2JDRA_L20
(AKT2)
CMGC
A-443654
I
44
255
61
44
255
61
A
2I0EA_PDS
(PRKCB)
CMGC
bisindolylma...
I
41
141
45
41
141
45
A
1NVRA_STU
(CHEK1)
CMGC
staurosporine
I
179
71
79
179
71
79
A
1SNUA_STU
(ITK)
CMGC
staurosporine
I
99
104
128
99
104
128
A
2XYNA_VX6
(ABL2)
CMGC
VX-680
I
79
101
105
79
101
105
A
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
62
139
51
A
3E5AA_VX6
(AURKA)
CMGC
VX-680
I
57
107
93
57
107
93
B
20
3MIYA_B49
(ITK)
CMGC
Sunitinib
I
70
74
110
B
3MIYA_B49
(ITK)
CMGC
Sunitinib
I
70
74
110
70
74
110
B
2PE2A_464
(PDPK1)
CMGC
Indolinone b...
I
134
156
104
134
156
104
B
3NYNA_SGV
(GRK6)
CMGC
SMR000127424
I
54
7
47
54
7
47
B
1UU9A_BI3
(PDPK1)
CMGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
3CD3A_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
2BMCA_MPY
(AURKA)
CMGC
PHA-680632
I
107
108
107
107
108
107
B
1UVRA_BI8
(PDPK1)
CMGC
Ro 31-7549
I
82
181
65
82
181
65
B
3ORZA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
3EFWA_AK8
(AURKA)
CMGC
3efw
I
100
59
105
100
59
105
B
3OTUA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
1ZRZA_BI1
(PRKCI)
CMGC
bisindolylma...
I
52
150
47
52
150
47
B
2C6EA_HPM
(AURKA)
CMGC
HPM
I
44
237
90
44
237
90
B
1UU7A_BI2
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
3BKBA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3L9MA_L9M
(PRKACA)
CMGC
VX_680
I
37
65
42
37
65
42
B
1UU8A_BI1
(PDPK1)
CMGC
bisindolylma...
I
83
189
65
83
189
65
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
1WVYA_STU
(DAPK1)
CMGC
staurosporine
I
83
23
55
83
23
55
B
3CBLA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138