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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
FER (
P16591
)
Kinase group
TK
Number of conformation types
0
Number of structural templates
68 (
Total 59 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
30
1AQ1A_STU
(CDK2)
TK
staurosporine
I
195
76
118
A
1AQ1A_STU
(CDK2)
TK
staurosporine
I
195
76
118
195
76
118
A
2DQ7X_STU
(FYN)
TK
staurosporine
I
91
74
124
91
74
124
A
1SM2A_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1XBCA_STU
(SYK)
TK
staurosporine
I
71
72
105
71
72
105
A
1XJDA_STU
(PRKCQ)
TK
staurosporine
I
121
101
106
121
101
106
A
1YVJA_4ST
(JAK3)
TK
staurosporine
I
96
90
126
96
90
126
A
3CKXA_STU
(STK24)
TK
staurosporine
I
176
104
141
176
104
141
A
1PKDA_UCN
(CDK2)
TK
UCN 02
I
195
67
118
195
67
118
A
2VTTA_LZD
(CDK2)
TK
pyrazole dia...
I
158
42
111
158
42
111
A
2IVUA_ZD6
(RET)
TK
Vandetanib
I
83
291
121
83
291
121
A
1R78A_FMD
(CDK2)
TK
4-alkynyl ox...
I
127
24
97
127
24
97
A
2H8HA_H8H
(SRC)
TK
Saracatinib
I
91
255
126
91
255
126
A
2IW6A_QQ2
(CDK2)
TK
2iw6
I
112
209
86
112
209
86
A
3EJ1A_5BP
(CDK2)
TK
AC1OCFRV
I
46
92
62
46
92
62
A
1OIYA_N41
(CDK2)
TK
N41
I
33
49
34
33
49
34
A
3PIYA_585
(BTK)
TK
R-406
I
93
17
123
93
17
123
A
2J51A_DKI
(SLK)
TK
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2IW8A_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
2WIHA_P48
(CDK2)
TK
VX_680
I
111
425
105
111
425
105
A
2JEDA_LG8
(PRKCQ)
TK
5-Arylidene-...
I
67
19
87
67
19
87
A
2JFLA_DKI
(SLK)
TK
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2IW9A_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
3PJ3A_04L
(BTK)
TK
Imatinib
II
99
113
134
99
113
134
A
1H1SA_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
3FQSA_585
(SYK)
TK
R-406
I
64
28
102
64
28
102
A
2R3NA_SCZ
(CDK2)
TK
AC1LZZHM
I
46
175
57
46
175
57
A
1OGUA_ST8
(CDK2)
TK
ST8
I
31
21
34
31
21
34
A
3LXLA_IZA
(JAK3)
TK
Pyridone 6
I
30
11
63
30
11
63
A
3IKAA_0UN
(EGFR)
TK
2jkk
I
76
120
108
76
120
108
B
36
3LCSA_STU
(ALK)
TK
staurosporine
I
73
100
109
B
3LCSA_STU
(ALK)
TK
staurosporine
I
73
100
109
73
100
109
B
2ITQA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
2ITUA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
2ITWA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
1WVYA_STU
(DAPK1)
TK
staurosporine
I
83
23
55
83
23
55
B
3BKBA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3MIYA_B49
(ITK)
TK
Sunitinib
I
70
74
110
70
74
110
B
2WKMA_PFY
(MET)
TK
PHA-665752
I
38
34
98
38
34
98
B
2X9FA_X9F
(EPHB4)
TK
X9F
I
46
19
86
46
19
86
B
3EFWA_AK8
(AURKA)
TK
3efw
I
100
59
105
100
59
105
B
2WTWA_ZZL
(AURKA)
TK
MLN8054
I
35
24
70
35
24
70
B
3H10A_97B
(AURKA)
TK
MLN8054
I
39
88
82
39
88
82
B
1H07A_MFP
(CDK2)
TK
AC1NAKJQ
I
90
241
80
90
241
80
B
2ITOA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITYA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITZA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
77
287
111
B
3F5PA_741
(IGF1R)
TK
3-cyanoquino...
I
60
123
81
60
123
81
B
3NZ0A_IZA
(TYK2)
TK
Pyridone 6
I
12
3
24
12
3
24
B
3NRMA_NRM
(AURKA)
TK
CAS404828_08_6
I
32
33
60
32
33
60
B
2C6IA_DT1
(CDK2)
TK
2c6i
I
27
41
48
27
41
48
B
3MTLA_FEF
(PCTK1)
TK
indirubin de...
I
16
3
23
16
3
23
B
2XB7A_GUI
(ALK)
TK
NVP-TAE684
I
71
66
107
71
66
107
B
3P9JA_P9J
(AURKA)
TK
4-[(5-Methyl...
I
32
50
54
32
50
54
B
2C6OA_4SP
(CDK2)
TK
nu6102
I
23
33
27
23
33
27
B
3EKNA_GS3
(INSR)
TK
pyrrolo[2,3-...
I
90
215
127
90
215
127
B
2BMCA_MPY
(AURKA)
TK
PHA-680632
I
107
108
107
107
108
107
B
3EKKA_GS2
(INSR)
TK
pyrrolo[2,3-...
I
33
131
65
33
131
65
B
3LW0A_CCX
(IGF1R)
TK
5-vinyl-3-py...
III
53
30
101
53
30
101
B
3COHA_83H
(AURKA)
TK
AKI-001
I
79
88
65
79
88
65
B
3AMAA_SKE
(PRKACA)
TK
JNJ-7706621
I
46
26
35
46
26
35
B
2B7AA_IZA
(JAK2)
TK
Pyridone 6
I
34
12
65
34
12
65
B
3FQEA_P5C
(SYK)
TK
AMG_706
I
24
88
63
24
88
63
B
3EYHA_IZA
(JAK1)
TK
Pyridone 6
I
21
19
54
21
19
54
D
2
1R0PA_KSA
(MET)
TK
k-252a
I
28
79
64
D
1R0PA_KSA
(MET)
TK
k-252a
I
28
79
64
28
79
64
D
2WGJA_VGH
(MET)
TK
Crizotinib
I
21
23
55
21
23
55