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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
LTK (
P29376
)
Kinase group
TK
Number of conformation types
0
Number of structural templates
57 (
Total 72 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
30
1QPJA_STU
(LCK)
TK
staurosporine
I
115
76
126
A
1QPJA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
1SM2A_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1U59A_STU
(ZAP70)
TK
staurosporine
I
96
80
114
96
80
114
A
1XBCA_STU
(SYK)
TK
staurosporine
I
71
72
105
71
72
105
A
1YVJA_4ST
(JAK3)
TK
staurosporine
I
96
90
126
96
90
126
A
3CKXA_STU
(STK24)
TK
staurosporine
I
176
104
141
176
104
141
A
1BYGA_STU
(CSK)
TK
staurosporine
I
85
72
123
85
72
123
A
2DQ7X_STU
(FYN)
TK
staurosporine
I
91
74
124
91
74
124
A
1QPDA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
2HZ4A_4ST
(ABL1)
TK
staurosporine
I
159
103
156
159
103
156
A
2IVUA_ZD6
(RET)
TK
Vandetanib
I
83
291
121
83
291
121
A
2H8HA_H8H
(SRC)
TK
Saracatinib
I
91
255
126
91
255
126
A
2C0IA_L1G
(HCK)
TK
A-420983
I
61
269
86
61
269
86
A
2C0TA_L3G
(HCK)
TK
A-641359
I
48
260
84
48
260
84
A
2OFUA_1N9
(LCK)
TK
2-aminopyrim...
I
55
215
101
55
215
101
A
1M17A_AQ4
(EGFR)
TK
Erlotinib
I
43
166
82
43
166
82
A
2F4JA_VX6
(ABL1)
TK
VX-680
I
110
109
134
110
109
134
A
2XYNA_VX6
(ABL2)
TK
VX-680
I
79
101
105
79
101
105
A
2X2MA_X2M
(RET)
TK
Semaxanib
I
24
81
59
24
81
59
A
3PJ3A_04L
(BTK)
TK
Imatinib
II
99
113
134
99
113
134
A
3LXLA_IZA
(JAK3)
TK
Pyridone 6
I
30
11
63
30
11
63
A
3FQSA_585
(SYK)
TK
R-406
I
64
28
102
64
28
102
A
1AGWA_SU2
(FGFR1)
TK
SU 4984
I
77
81
111
77
81
111
A
3LXPA_IZA
(TYK2)
TK
Pyridone 6
I
9
3
20
9
3
20
A
3IKAA_0UN
(EGFR)
TK
2jkk
I
76
120
108
76
120
108
A
2C0OA_L2G
(HCK)
TK
A-770041
I
41
222
65
41
222
65
A
3PIYA_585
(BTK)
TK
R-406
I
93
17
123
93
17
123
A
1FGIA_SU1
(FGFR1)
TK
Indolin-2-on...
I
25
71
61
25
71
61
A
2X2KA_X2K
(RET)
TK
Semaxanib
I
23
30
58
23
30
58
B
23
3LCSA_STU
(ALK)
TK
staurosporine
I
73
100
109
B
3LCSA_STU
(ALK)
TK
staurosporine
I
73
100
109
73
100
109
B
2ITQA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
2ITUA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
2ITWA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
3BKBA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3MIYA_B49
(ITK)
TK
Sunitinib
I
70
74
110
70
74
110
B
3D7TA_STU
(CSK)
TK
staurosporine
I
70
68
99
70
68
99
B
2ITOA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITYA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITZA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
77
287
111
B
2WKMA_PFY
(MET)
TK
PHA-665752
I
38
34
98
38
34
98
B
3AOXA_EMH
(ALK)
TK
BIRB_796
I
34
28
85
34
28
85
B
3EKKA_GS2
(INSR)
TK
pyrrolo[2,3-...
I
33
131
65
33
131
65
B
3EKNA_GS3
(INSR)
TK
pyrrolo[2,3-...
I
90
215
127
90
215
127
B
2B7AA_IZA
(JAK2)
TK
Pyridone 6
I
34
12
65
34
12
65
B
3EYHA_IZA
(JAK1)
TK
Pyridone 6
I
21
19
54
21
19
54
B
2X9FA_X9F
(EPHB4)
TK
X9F
I
46
19
86
46
19
86
B
3NZ0A_IZA
(TYK2)
TK
Pyridone 6
I
12
3
24
12
3
24
B
3F5PA_741
(IGF1R)
TK
3-cyanoquino...
I
60
123
81
60
123
81
B
2XB7A_GUI
(ALK)
TK
NVP-TAE684
I
71
66
107
71
66
107
D
4
1R0PA_KSA
(MET)
TK
k-252a
I
28
79
64
D
1R0PA_KSA
(MET)
TK
k-252a
I
28
79
64
28
79
64
D
3A4PA_DFQ
(MET)
TK
EKB_569
I
2
17
8
2
17
8
D
2RFSA_AM8
(MET)
TK
SU11274
I
7
3
35
7
3
35
D
2WGJA_VGH
(MET)
TK
Crizotinib
I
21
23
55
21
23
55