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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
RPS6KA4 (
O75676
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
15 (
Total 69 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
15
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
2JAMA_J60
(CAMK1G)
AGC
SU11652
I
50
65
32
50
65
32
A
1R78A_FMD
(CDK2)
AGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
2VTTA_LZD
(CDK2)
AGC
pyrazole dia...
I
158
42
111
158
42
111
A
1OI9A_N20
(CDK2)
AGC
NU-6086
I
52
80
61
52
80
61
A
2J51A_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2JFLA_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
3NLBA_5BE
(CHEK1)
AGC
38P
I
45
115
49
45
115
49
A
2J90A_IZA
(DAPK3)
AGC
Pyridone 6
I
40
50
42
40
50
42
A
2I40A_BLZ
(CDK2)
AGC
2i40
I
34
95
16
34
95
16
A
2E9VA_85A
(CHEK1)
AGC
macrocyclic ...
I
14
121
27
14
121
27