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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
P48
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
CDK2 (PDB code: 2WIH)
[PDB]
[PDBsum]
Inhibitor
VX_680 (HET code: P48)
[PDB]
Summary of KIF 2WIHA_P48
(CDK2, PDB code:
2WIH
, chain A)
Number of family interactions
953
Number of family kinase
111 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
425 (1 are CDKL3 inhibitors)
Involved diseases
105 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
CDKL3 and 1 inhibitors