Protein Surface  Ribbon
Inhibitor X8E
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase CHEK1 (PDB code: 2X8E) [PDB] [PDBsum]
Inhibitor CAS318480_82_9 (HET code: X8E) [PDB]
 
Summary of KIF 2X8EA_X8E (CHEK1, PDB code: 2X8E, chain A)
Number of family interactions 31
Number of family kinase 4 (sequence conservation) (profiling results)
Number of family inhibitors 31 (22 are CHEK1 inhibitors)
Involved diseases 16 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  CHEK1 and 22 inhibitors