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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
J60
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
STK25 (PDB code: 2XIK)
[PDB]
[PDBsum]
Inhibitor
SU11652 (HET code: J60)
[PDB]
Summary of KIF 2XIKA_J60
(STK25, PDB code:
2XIK
, chain A)
Number of family interactions
426
Number of family kinase
59 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
49 (4 are GRK4 inhibitors)
Involved diseases
65 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
GRK4 and 4 inhibitors