Protein Surface  Ribbon
Inhibitor 877
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase MAPK8 (PDB code: 2GMX) [PDB] [PDBsum]
Inhibitor N-(4-AMINO-5-CYANO-6-ETHOXYPYRIDIN-2-YL)-2-(4-BROMO-2,5-DIMETHOXYPHENYL)ACETAMIDE (HET code: 877) [PDB]
 
Summary of KIF 2GMXA_877 (MAPK8, PDB code: 2GMX, chain A)
Number of family interactions 56
Number of family kinase 3 (sequence conservation) (profiling results)
Number of family inhibitors 29 (29 are MAPK8 inhibitors)
Involved diseases 14 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  MAPK8 and 29 inhibitors