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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
DKI
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
CLK3 (PDB code: 2WU6)
[PDB]
[PDBsum]
Inhibitor
5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE (HET code: DKI)
[PDB]
Summary of KIF 2WU6A_DKI
(CLK3, PDB code:
2WU6
, chain A)
Number of family interactions
77
Number of family kinase
26 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
9 (1 are NLK inhibitors)
Involved diseases
26 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
NLK and 1 inhibitors