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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
IZA
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
JAK2 (PDB code: 2B7A)
[PDB]
[PDBsum]
Inhibitor
Pyridone 6 (HET code: IZA)
[PDB]
Summary of KIF 2B7AA_IZA
(JAK2, PDB code:
2B7A
, chain A)
Number of family interactions
46
Number of family kinase
34 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
12 (1 are NTRK1 inhibitors)
Involved diseases
65 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
NTRK1 and 1 inhibitors