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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
TAK
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
ACVR1 (PDB code: 3H9R)
[PDB]
[PDBsum]
Inhibitor
dorsomorphin (HET code: TAK)
[PDB]
Summary of KIF 3H9RA_TAK
(ACVR1, PDB code:
3H9R
, chain A)
Number of family interactions
96
Number of family kinase
15 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
67 (1 are TGFBR2 inhibitors)
Involved diseases
37 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
TGFBR2 and 1 inhibitors