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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
VX6
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
AURKA (PDB code: 3E5A)
[PDB]
[PDBsum]
Inhibitor
VX-680 (HET code: VX6)
[PDB]
Summary of KIF 3E5AA_VX6
(AURKA, PDB code:
3E5A
, chain A)
Number of family interactions
357
Number of family kinase
57 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
107 (2 are TNK1 inhibitors)
Involved diseases
93 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
TNK1 and 2 inhibitors