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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
MI1
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
JAK1 (PDB code: 3EYG)
[PDB]
[PDBsum]
Inhibitor
CP690550 (HET code: MI1)
[PDB]
Summary of KIF 3EYGA_MI1
(JAK1, PDB code:
3EYG
, chain A)
Number of family interactions
55
Number of family kinase
8 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
23 (2 are TNK1 inhibitors)
Involved diseases
31 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
TNK1 and 2 inhibitors