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Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
MI1
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
JAK2 (PDB code: 3FUP)
[PDB]
[PDBsum]
Inhibitor
CP690550 (HET code: MI1)
[PDB]
Summary of KIF 3FUPA_MI1
(JAK2, PDB code:
3FUP
, chain A)
Number of family interactions
76
Number of family kinase
16 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
27 (2 are TNK1 inhibitors)
Involved diseases
32 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
TNK1 and 2 inhibitors