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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
1 PIM1 related diseases
hsa05221
Acute myeloid leukemia
Summary of query kinase
Query kinase
PIM3 (
Q86V86
),
reference kinase: PIM1
(
P11309
)
Kinase group
CAMK
Number of conformation types
2
Number of structural templates
50 (
Total 392 inhibitors
)
Number of PIM1 related diseases
1 (
hsa05221
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
48
1YHSA_STU
(PIM1)
CAMK
staurosporine
I
78
64
50
A
1YHSA_STU
(PIM1)
CAMK
staurosporine
I
78
64
50
78
64
50
A
1XWSA_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
2BILB_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
2BIKB_BI1
(PIM1)
CAMK
bisindolylma...
I
41
132
36
41
132
36
A
2J2IB_LY4
(PIM1)
CAMK
Ruboxistaurin
I
35
89
36
35
89
36
A
2BZKB_ANP
(PIM1)
CAMK
Phosphoamino...
I
14
7
23
14
7
23
A
1XR1A_ANP
(PIM1)
CAMK
Phosphoamino...
I
14
7
23
14
7
23
A
1YXUA_AMP
(PIM1)
CAMK
Adenosine mo...
I
14
9
23
14
9
23
A
3A99A_ANP
(PIM1)
CAMK
Phosphoamino...
I
14
7
23
14
7
23
A
3BGQA_VX2
(PIM1)
CAMK
triazolopyri...
I
10
25
14
10
25
14
A
3BGZA_VX3
(PIM1)
CAMK
2,3-diphenyl...
I
9
14
8
9
14
8
A
3CY2A_MB9
(PIM1)
CAMK
AT_7519
I
8
7
16
8
7
16
A
3CY3A_JN5
(PIM1)
CAMK
JN5
I
8
10
10
8
10
10
A
1YI4A_ADN
(PIM1)
CAMK
Vidarabine
I
7
8
10
7
8
10
A
2O63A_MYC
(PIM1)
CAMK
quercetin
I
5
25
8
5
25
8
A
2O3PA_QUE
(PIM1)
CAMK
quercetin
I
5
25
8
5
25
8
A
3JPVA_1DR
(PIM1)
CAMK
1DR
I
5
11
2
5
11
2
A
3BWFA_DWC
(PIM1)
CAMK
HB12
I
4
9
2
4
9
2
A
3JXWA_LXG
(PIM1)
CAMK
benzothienop...
I
4
19
2
4
19
2
A
3JYAA_LWG
(PIM1)
CAMK
Kinome_3259
I
4
5
1
4
5
1
A
3R04A_UNQ
(PIM1)
CAMK
5-{6-[(Trans...
I
4
21
4
4
21
4
A
2O64A_MYU
(PIM1)
CAMK
Quercetagetin
I
4
24
7
4
24
7
A
2BZIB_DW2
(PIM1)
CAMK
HB12
I
4
9
2
4
9
2
A
2C3IB_IYZ
(PIM1)
CAMK
AC1NURHU
I
4
12
2
4
12
2
A
2O65A_MYF
(PIM1)
CAMK
luteolin
I
4
24
7
4
24
7
A
3CXWA_7CP
(PIM1)
CAMK
AT_7519
I
3
5
1
3
5
1
A
3DCVA_55E
(PIM1)
CAMK
ZINC13780154
I
3
3
12
3
3
12
A
3F2AA_985
(PIM1)
CAMK
pyrazine inh...
I
3
16
1
3
16
1
A
1YI3A_LY2
(PIM1)
CAMK
LY294002
I
3
2
2
3
2
2
A
2XJ2A_985
(PIM1)
CAMK
pyrazine inh...
I
3
16
1
3
16
1
A
2XJ1A_XJ1
(PIM1)
CAMK
pyrazine inh...
I
3
26
1
3
26
1
A
3JY0A_LYG
(PIM1)
CAMK
benzothienop...
I
2
16
1
2
16
1
A
3MA3A_01I
(PIM1)
CAMK
AC1LAPMW
I
2
2
4
2
2
4
A
3QF9A_NM8
(PIM1)
CAMK
AC1O76GQ
I
2
2
6
2
2
6
A
3R02A_UNM
(PIM1)
CAMK
7-[(Cis-4-Am...
I
2
13
1
2
13
1
A
2BZHB_HB1
(PIM1)
CAMK
HB12
I
2
4
1
2
4
1
A
2BZJA_ME3
(PIM1)
CAMK
BSQFHYQBCYIA...
I
2
4
2
2
4
2
A
3C4EA_C4E
(PIM1)
CAMK
Phenyl-quina...
I
2
2
2
2
2
2
A
2OBJA_VRV
(PIM1)
CAMK
2obj
I
2
10
2
2
10
2
A
2OI4X_JM1
(PIM1)
CAMK
HB12
I
2
4
1
2
4
1
A
2XIYA_XIY
(PIM1)
CAMK
6-methoxyqui...
I
1
1
1
1
1
1
A
3R01A_UNE
(PIM1)
CAMK
5-bromo-7-me...
I
1
5
1
1
5
1
A
3R00A_UNJ
(PIM1)
CAMK
5-bromo-1-be...
I
1
5
1
1
5
1
A
2XJ0A_XJ0
(PIM1)
CAMK
7,8-dihydro-...
I
1
1
1
1
1
1
A
1YXVA_LI6
(PIM1)
CAMK
AC1NSQEB
I
1
1
1
1
1
1
A
1YXXA_LI7
(PIM1)
CAMK
DNC010328
I
1
1
1
1
1
1
A
3BGPA_VX1
(PIM1)
CAMK
3bgp
I
1
2
1
1
2
1
A
2XIXA_XIX
(PIM1)
CAMK
XIX
I
1
1
1
1
1
1
B
2
1YXTA_ANP
(PIM1)
CAMK
Phosphoamino...
I
14
6
21
B
1YXTA_ANP
(PIM1)
CAMK
Phosphoamino...
I
14
6
21
14
6
21
B
2XIZA_XIZ
(PIM1)
CAMK
Phenylmaloni...
I
1
1
1
1
1
1