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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
RPS6KA6 (
Q9UK32
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
76 (
Total 90 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
64
1Q3DA_STU
(GSK3B)
AGC
staurosporine
I
115
71
61
A
1Q3DA_STU
(GSK3B)
AGC
staurosporine
I
115
71
61
115
71
61
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
1SM2A_STU
(ITK)
AGC
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
AGC
staurosporine
I
99
104
128
99
104
128
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
1YHSA_STU
(PIM1)
AGC
staurosporine
I
78
64
50
78
64
50
A
1NXKA_STU
(MAPKAPK2)
AGC
staurosporine
I
110
67
51
110
67
51
A
2HZ4A_4ST
(ABL1)
AGC
staurosporine
I
159
103
156
159
103
156
A
3HMOA_STU
(TTK)
AGC
staurosporine
I
27
50
20
27
50
20
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
2BILB_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2OW3A_BIM
(GSK3B)
AGC
LY_333531
I
62
139
51
62
139
51
A
1XWSA_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2BIKB_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2J2IB_LY4
(PIM1)
AGC
Ruboxistaurin
I
35
89
36
35
89
36
A
2VTTA_LZD
(CDK2)
AGC
pyrazole dia...
I
158
42
111
158
42
111
A
3M2WA_L8I
(MAPKAPK2)
AGC
Sunitinib
I
84
90
47
84
90
47
A
2IVUA_ZD6
(RET)
AGC
Vandetanib
I
83
291
121
83
291
121
A
3BLRA_CPB
(CDK9)
AGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
2H8HA_H8H
(SRC)
AGC
Saracatinib
I
91
255
126
91
255
126
A
1A9UA_SB2
(MAPK14)
AGC
SB 203580
I
21
31
28
21
31
28
A
3GFWA_S22
(TTK)
AGC
1-(4-(4-(2-(...
I
21
4
18
21
4
18
A
1PMEA_SB2
(MAPK1)
AGC
SB 203580
I
16
31
26
16
31
26
A
1R78A_FMD
(CDK2)
AGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
3OBGA_SB2
(MAPK14)
AGC
SB 203580
I
21
31
28
21
31
28
A
2V7OA_DRN
(CAMK2G)
AGC
bisindolylma...
I
23
51
16
23
51
16
A
2X2MA_X2M
(RET)
AGC
Semaxanib
I
24
81
59
24
81
59
A
1Q3WA_ATU
(GSK3B)
AGC
alsterpaullone
I
24
28
19
24
28
19
A
1BL6A_SB6
(MAPK14)
AGC
sb216995
I
46
110
50
46
110
50
A
2J51A_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2JFLA_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2C0OA_L2G
(HCK)
AGC
A-770041
I
41
222
65
41
222
65
A
2X2KA_X2K
(RET)
AGC
Semaxanib
I
23
30
58
23
30
58
A
1H1SA_4SP
(CDK2)
AGC
nu6102
I
30
33
30
30
33
30
A
3PA5A_C73
(CHEK1)
AGC
2-(Carbamoyl...
I
15
74
20
15
74
20
A
3L8XA_N4D
(MAPK14)
AGC
3cg2
I
91
104
65
91
104
65
A
1OZ1A_FPH
(MAPK14)
AGC
4-Azaindole 6
I
18
27
28
18
27
28
A
3H9FA_92M
(TTK)
AGC
Mps1-IN-2
I
12
7
6
12
7
6
A
1OGUA_ST8
(CDK2)
AGC
ST8
I
31
21
34
31
21
34
A
2WELA_K88
(CAMK2D)
AGC
su6656
I
30
30
15
30
30
15
A
3PJ3A_04L
(BTK)
AGC
Imatinib
II
99
113
134
99
113
134
A
3FKOA_FKO
(MAPK14)
AGC
L-779450
I
17
7
27
17
7
27
A
3MVLA_38P
(MAPK14)
AGC
38P
I
50
308
44
50
308
44
A
1OIYA_N41
(CDK2)
AGC
N41
I
33
49
34
33
49
34
A
1UV5A_BRW
(GSK3B)
AGC
6-bromoindir...
I
27
37
28
27
37
28
A
2IW6A_QQ2
(CDK2)
AGC
2iw6
I
112
209
86
112
209
86
A
1QCFA_PP1
(HCK)
AGC
PP1
I
31
65
68
31
65
68
A
2Z7SA_P01
(RPS6KA1)
AGC
Lopac0_000938
I
32
214
49
32
214
49
A
2IW8A_4SP
(CDK2)
AGC
nu6102
I
30
33
30
30
33
30
A
2BHEA_BRY
(CDK2)
AGC
BRY
I
51
31
35
51
31
35
A
2IVVA_PP1
(RET)
AGC
PP1
I
27
46
63
27
46
63
A
3DOGA_NNN
(CDK2)
AGC
NSC743927
I
50
239
48
50
239
48
A
2IW9A_4SP
(CDK2)
AGC
nu6102
I
30
33
30
30
33
30
A
2I40A_BLZ
(CDK2)
AGC
2i40
I
34
95
16
34
95
16
A
2ZB1A_GK4
(MAPK14)
AGC
biphenyl ami...
II
55
57
54
55
57
54
A
3HA8A_5JZ
(MAPK14)
AGC
DEL-B, 14b
I
59
89
62
59
89
62
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
1ZZLA_TZY
(MAPK14)
AGC
CP-808844
I
36
84
44
36
84
44
A
3E92A_G6A
(MAPK14)
AGC
3e92
I
56
59
55
56
59
55
A
2C0IA_L1G
(HCK)
AGC
A-420983
I
61
269
86
61
269
86
A
3NLBA_5BE
(CHEK1)
AGC
38P
I
45
115
49
45
115
49
A
2J90A_IZA
(DAPK3)
AGC
Pyridone 6
I
40
50
42
40
50
42
A
3IPHA_G11
(MAPK14)
AGC
HMS3303K05
I
57
108
55
57
108
55
B
12
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
52
150
47
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
2PE2A_464
(PDPK1)
AGC
Indolinone b...
I
134
156
104
134
156
104
B
1UNLA_RRC
(CDK5)
AGC
roscovitine
I
45
237
47
45
237
47