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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
4 CDKL5 related diseases
H00478
Prader-Willi and Angelman syndromes
H00606
Early infantile epileptic encephalopathy
105830
Angelman syndrome-like
300672
Epileptic encephalopathy, early infantile, 2
Summary of query kinase
Query kinase
CDKL5 (
O76039
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
44 (
Total 13 inhibitors
)
Number of CDKL5 related diseases
4 (
H00478
H00606
105830
300672
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
31
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
A
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
121
101
106
A
2F4JA_VX6
(ABL1)
CMGC
VX-680
I
110
109
134
110
109
134
A
2BILB_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1YHSA_STU
(PIM1)
CMGC
staurosporine
I
78
64
50
78
64
50
A
2WIHA_P48
(CDK2)
CMGC
VX_680
I
111
425
105
111
425
105
A
2I0EA_PDS
(PRKCB)
CMGC
bisindolylma...
I
41
141
45
41
141
45
A
1NVQA_UCN
(CHEK1)
CMGC
UCN 02
I
179
65
79
179
65
79
A
2HY81_1ST
(PAK1)
CMGC
UCN 02
I
58
20
75
58
20
75
A
2XYNA_VX6
(ABL2)
CMGC
VX-680
I
79
101
105
79
101
105
A
2VTQA_LZA
(CDK2)
CMGC
pyrazole dia...
I
36
25
31
36
25
31
A
2J2IB_LY4
(PIM1)
CMGC
Ruboxistaurin
I
35
89
36
35
89
36
A
1NVRA_STU
(CHEK1)
CMGC
staurosporine
I
179
71
79
179
71
79
A
2HZ4A_4ST
(ABL1)
CMGC
staurosporine
I
159
103
156
159
103
156
A
3E5AA_VX6
(AURKA)
CMGC
VX-680
I
57
107
93
57
107
93
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
A
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
62
139
51
A
1NXKA_STU
(MAPKAPK2)
CMGC
staurosporine
I
110
67
51
110
67
51
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
2VU3A_LZE
(CDK2)
CMGC
AT7519
I
35
22
29
35
22
29
A
3IW4A_LW4
(PRKCA)
CMGC
Sotrastaurin
I
52
119
49
52
119
49
A
3FMEA_STU
(MAP2K6)
CMGC
staurosporine
I
28
15
20
28
15
20
A
3M2WA_L8I
(MAPKAPK2)
CMGC
Sunitinib
I
84
90
47
84
90
47
A
1XWSA_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
3HMOA_STU
(TTK)
CMGC
staurosporine
I
27
50
20
27
50
20
A
2JDRA_L20
(AKT2)
CMGC
A-443654
I
44
255
61
44
255
61
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
3GFWA_S22
(TTK)
CMGC
1-(4-(4-(2-(...
I
21
4
18
21
4
18
A
3BLRA_CPB
(CDK9)
CMGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
2BIKB_BI1
(PIM1)
CMGC
bisindolylma...
I
41
132
36
41
132
36
B
13
3NYNA_SGV
(GRK6)
CMGC
SMR000127424
I
54
7
47
B
3NYNA_SGV
(GRK6)
CMGC
SMR000127424
I
54
7
47
54
7
47
B
1UU3A_LY4
(PDPK1)
CMGC
Ruboxistaurin
I
71
117
57
71
117
57
B
3EFWA_AK8
(AURKA)
CMGC
3efw
I
100
59
105
100
59
105
B
1UU7A_BI2
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
CMGC
bisindolylma...
I
83
189
65
83
189
65
B
1UU9A_BI3
(PDPK1)
CMGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
CMGC
Ro 31-7549
I
82
181
65
82
181
65
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
3ORZA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
1ZRZA_BI1
(PRKCI)
CMGC
bisindolylma...
I
52
150
47
52
150
47
B
3OTUA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
2FVDA_LIA
(CDK2)
CMGC
[4-Amino-2-[...
I
39
16
29
39
16
29