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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
EPHB3 (
P54753
)
Kinase group
TK
Number of conformation types
0
Number of structural templates
32 (
Total 37 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
18
2GQGA_1N1
(ABL1)
TK
Dasatinib
I
74
32
117
A
2GQGA_1N1
(ABL1)
TK
Dasatinib
I
74
32
117
74
32
117
A
3K54A_1N1
(BTK)
TK
Dasatinib
I
56
32
103
56
32
103
A
3OCTA_1N1
(BTK)
TK
Dasatinib
I
56
32
103
56
32
103
A
2VTQA_LZA
(CDK2)
TK
pyrazole dia...
I
36
25
31
36
25
31
A
2VU3A_LZE
(CDK2)
TK
AT7519
I
35
22
29
35
22
29
A
2H8HA_H8H
(SRC)
TK
Saracatinib
I
91
255
126
91
255
126
A
2VTTA_LZD
(CDK2)
TK
pyrazole dia...
I
158
42
111
158
42
111
A
2IW6A_QQ2
(CDK2)
TK
2iw6
I
112
209
86
112
209
86
A
3RHXA_3RH
(FGFR1)
TK
6-o-tolylqui...
I
27
31
67
27
31
67
A
3RI1A_3RH
(FGFR2)
TK
6-o-tolylqui...
I
29
33
72
29
33
72
A
1OPLA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
2FO0A_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
3L8XA_N4D
(MAPK14)
TK
3cg2
I
91
104
65
91
104
65
A
2G2HA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
1QCFA_PP1
(HCK)
TK
PP1
I
31
65
68
31
65
68
A
2HZIA_JIN
(ABL1)
TK
PD180970
I
90
77
120
90
77
120
A
1QPEA_PP2
(LCK)
TK
AG 1879
I
29
63
51
29
63
51
A
1WZYA_F29
(MAPK1)
TK
AC1O4W7N
I
27
48
33
27
48
33
B
14
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
B
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
77
287
111
B
2J5FA_DJK
(EGFR)
TK
4-anilinoqui...
I
16
212
45
16
212
45
B
3F5PA_741
(IGF1R)
TK
3-cyanoquino...
I
60
123
81
60
123
81
B
1H07A_MFP
(CDK2)
TK
AC1NAKJQ
I
90
241
80
90
241
80
B
2ITOA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2VTLA_LZ5
(CDK2)
TK
MLS000519301
I
5
18
17
5
18
17
B
2ITYA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2VTOA_LZ8
(CDK2)
TK
pyrazole dia...
I
10
26
27
10
26
27
B
2ITZA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2VTPA_LZ9
(CDK2)
TK
pyrazole dia...
I
6
18
17
6
18
17
B
2W1HA_L0H
(CDK2)
TK
DB08066
I
20
43
42
20
43
42
B
2VX1A_7X8
(EPHB4)
TK
DB07256
I
19
37
15
19
37
15
B
2XB7A_GUI
(ALK)
TK
NVP-TAE684
I
71
66
107
71
66
107
B
3EKNA_GS3
(INSR)
TK
pyrrolo[2,3-...
I
90
215
127
90
215
127