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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
MAP3K10 (
Q02779
)
Kinase group
TKL
Number of conformation types
0
Number of structural templates
15 (
Total 55 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
15
3EQFA_KSA
(MAP2K1)
TKL
k-252a
I
42
51
57
A
3EQFA_KSA
(MAP2K1)
TKL
k-252a
I
42
51
57
42
51
57
A
3CKXA_STU
(STK24)
TKL
staurosporine
I
176
104
141
176
104
141
A
1AQ1A_STU
(CDK2)
TKL
staurosporine
I
195
76
118
195
76
118
A
1SM2A_STU
(ITK)
TKL
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
TKL
staurosporine
I
99
104
128
99
104
128
A
1PKDA_UCN
(CDK2)
TKL
UCN 02
I
195
67
118
195
67
118
A
2WIHA_P48
(CDK2)
TKL
VX_680
I
111
425
105
111
425
105
A
3DTCA_VIN
(MAP3K9)
TKL
CEP-6331
I
6
21
16
6
21
16
A
1VYWA_292
(CDK2)
TKL
PNU-292137 I...
I
20
91
38
20
91
38
A
2IW6A_QQ2
(CDK2)
TKL
2iw6
I
112
209
86
112
209
86
A
1H1SA_4SP
(CDK2)
TKL
nu6102
I
30
33
30
30
33
30
A
1OGUA_ST8
(CDK2)
TKL
ST8
I
31
21
34
31
21
34
A
1OIYA_N41
(CDK2)
TKL
N41
I
33
49
34
33
49
34
A
2IW8A_4SP
(CDK2)
TKL
nu6102
I
30
33
30
30
33
30
A
2IW9A_4SP
(CDK2)
TKL
nu6102
I
30
33
30
30
33
30