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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
PRKD1 (
Q15139
)
Kinase group
CAMK
Number of conformation types
0
Number of structural templates
81 (
Total 67 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
54
2JAMA_J60
(CAMK1G)
CAMK
SU11652
I
50
65
32
A
2JAMA_J60
(CAMK1G)
CAMK
SU11652
I
50
65
32
50
65
32
A
2HZ4A_4ST
(ABL1)
CAMK
staurosporine
I
159
103
156
159
103
156
A
1Q3DA_STU
(GSK3B)
CAMK
staurosporine
I
115
71
61
115
71
61
A
3A4OX_STU
(LYN)
CAMK
staurosporine
I
73
70
88
73
70
88
A
1AQ1A_STU
(CDK2)
CAMK
staurosporine
I
195
76
118
195
76
118
A
1U59A_STU
(ZAP70)
CAMK
staurosporine
I
96
80
114
96
80
114
A
1NVRA_STU
(CHEK1)
CAMK
staurosporine
I
179
71
79
179
71
79
A
1XJDA_STU
(PRKCQ)
CAMK
staurosporine
I
121
101
106
121
101
106
A
1NXKA_STU
(MAPKAPK2)
CAMK
staurosporine
I
110
67
51
110
67
51
A
1YHSA_STU
(PIM1)
CAMK
staurosporine
I
78
64
50
78
64
50
A
3CKXA_STU
(STK24)
CAMK
staurosporine
I
176
104
141
176
104
141
A
2HW7A_STU
(MKNK2)
CAMK
staurosporine
I
28
55
16
28
55
16
A
2HY81_1ST
(PAK1)
CAMK
UCN 02
I
58
20
75
58
20
75
A
3M2WA_L8I
(MAPKAPK2)
CAMK
Sunitinib
I
84
90
47
84
90
47
A
1PKDA_UCN
(CDK2)
CAMK
UCN 02
I
195
67
118
195
67
118
A
1NVQA_UCN
(CHEK1)
CAMK
UCN 02
I
179
65
79
179
65
79
A
2J7TA_274
(STK10)
CAMK
SU11274
I
66
20
77
66
20
77
A
2JAVA_5Z5
(NEK2)
CAMK
pyrrollylact...
I
25
40
24
25
40
24
A
2VTTA_LZD
(CDK2)
CAMK
pyrazole dia...
I
158
42
111
158
42
111
A
2J51A_DKI
(SLK)
CAMK
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
1R78A_FMD
(CDK2)
CAMK
4-alkynyl ox...
I
127
24
97
127
24
97
A
2JFLA_DKI
(SLK)
CAMK
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
1WZYA_F29
(MAPK1)
CAMK
AC1O4W7N
I
27
48
33
27
48
33
A
3FYKX_B98
(MAPKAPK2)
CAMK
DB07431
I
4
20
0
4
20
0
A
1YI4A_ADN
(PIM1)
CAMK
Vidarabine
I
7
8
10
7
8
10
A
3KB7A_071
(PLK1)
CAMK
MLN_518
I
39
176
54
39
176
54
A
3PA4A_C72
(CHEK1)
CAMK
2-(4-Chlorop...
I
10
79
24
10
79
24
A
3PJ3A_04L
(BTK)
CAMK
Imatinib
II
99
113
134
99
113
134
A
3GU8A_3GU
(DAPK1)
CAMK
Vidarabine
I
14
17
24
14
17
24
A
3M42A_HGF
(MAPKAPK2)
CAMK
SB_431542
I
5
61
9
5
61
9
A
3MVLA_38P
(MAPK14)
CAMK
38P
I
50
308
44
50
308
44
A
2JBOA_P4O
(MAPKAPK2)
CAMK
2jbo
I
18
130
30
18
130
30
A
2IW6A_QQ2
(CDK2)
CAMK
2iw6
I
112
209
86
112
209
86
A
3BHHA_5CP
(CAMK2B)
CAMK
DCL001071
I
17
45
22
17
45
22
A
2JBPA_P4O
(MAPKAPK2)
CAMK
2jbo
I
18
130
30
18
130
30
A
1PMVA_537
(MAPK10)
CAMK
1,9-Pyrazolo...
I
10
5
23
10
5
23
A
3D0EA_G93
(AKT2)
CAMK
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
3LM0A_EBD
(STK17B)
CAMK
DCL001071
I
20
106
24
20
106
24
A
3DS6A_A17
(MAPK14)
CAMK
3ds6
II
21
146
34
21
146
34
A
2JEDA_LG8
(PRKCQ)
CAMK
5-Arylidene-...
I
67
19
87
67
19
87
A
1UKIA_537
(MAPK8)
CAMK
1,9-Pyrazolo...
I
20
4
24
20
4
24
A
1BL6A_SB6
(MAPK14)
CAMK
sb216995
I
46
110
50
46
110
50
A
2ZB1A_GK4
(MAPK14)
CAMK
biphenyl ami...
II
55
57
54
55
57
54
A
2O0UA_C0M
(MAPK10)
CAMK
ZINC00799686
I
21
8
23
21
8
23
A
1NVSA_UCM
(CHEK1)
CAMK
SB218078
I
97
6
53
97
6
53
A
1ZZLA_TZY
(MAPK14)
CAMK
CP-808844
I
36
84
44
36
84
44
A
3E92A_G6A
(MAPK14)
CAMK
3e92
I
56
59
55
56
59
55
A
2RKUA_R78
(PLK1)
CAMK
BI 2536
I
37
59
35
37
59
35
A
2J90A_IZA
(DAPK3)
CAMK
Pyridone 6
I
40
50
42
40
50
42
A
3IPHA_G11
(MAPK14)
CAMK
HMS3303K05
I
57
108
55
57
108
55
A
3R2YA_P4O
(MAPKAPK2)
CAMK
2jbo
I
18
130
30
18
130
30
A
3FC2A_IBI
(PLK1)
CAMK
BI 2536
I
38
72
42
38
72
42
A
3PA3A_C70
(CHEK1)
CAMK
2-(4-Chlorop...
I
11
72
16
11
72
16
A
3L8XA_N4D
(MAPK14)
CAMK
3cg2
I
91
104
65
91
104
65
B
27
3BKBA_STU
(FES)
CAMK
staurosporine
I
131
107
138
B
3BKBA_STU
(FES)
CAMK
staurosporine
I
131
107
138
131
107
138
B
1WVYA_STU
(DAPK1)
CAMK
staurosporine
I
83
23
55
83
23
55
B
3CBLA_STU
(FES)
CAMK
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
CAMK
staurosporine
I
131
107
138
131
107
138
B
2PE2A_464
(PDPK1)
CAMK
Indolinone b...
I
134
156
104
134
156
104
B
1OKYA_STU
(PDPK1)
CAMK
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CAMK
UCN 02
I
179
60
109
179
60
109
B
3EFWA_AK8
(AURKA)
CAMK
3efw
I
100
59
105
100
59
105
B
3NYNA_SGV
(GRK6)
CAMK
SMR000127424
I
54
7
47
54
7
47
B
3AMAA_SKE
(PRKACA)
CAMK
JNJ-7706621
I
46
26
35
46
26
35
B
3FZ1A_B98
(CDK2)
CAMK
DB07431
I
5
19
5
5
19
5
B
2VWUA_7X1
(EPHB4)
CAMK
Chlorobenzod...
I
77
287
111
77
287
111
B
2WTCA_VGM
(CHEK2)
CAMK
VGM
I
10
39
19
10
39
19
B
3PY0A_SU9
(CDK2)
CAMK
SU 9516
I
25
19
33
25
19
33
B
1H07A_MFP
(CDK2)
CAMK
AC1NAKJQ
I
90
241
80
90
241
80
B
3PY1A_SU9
(CDK2)
CAMK
SU 9516
I
25
19
33
25
19
33
B
2VTSA_LZC
(CDK2)
CAMK
DB08140
I
28
54
26
28
54
26
B
1H00A_FAP
(CDK2)
CAMK
AC1NAE4F
I
50
94
75
50
94
75
B
3CQWA_CQW
(AKT1)
CAMK
3cqw
I
3
8
23
3
8
23
B
2BMCA_MPY
(AURKA)
CAMK
PHA-680632
I
107
108
107
107
108
107
B
1P4FA_DRG
(DAPK1)
CAMK
benzopyrazol...
I
7
6
29
7
6
29
B
3FHRA_P4O
(MAPKAPK3)
CAMK
2jbo
I
17
110
31
17
110
31
B
3GOKA_P4O
(MAPKAPK2)
CAMK
2jbo
I
20
134
35
20
134
35
B
3COHA_83H
(AURKA)
CAMK
AKI-001
I
79
88
65
79
88
65
B
1MUOA_ADN
(AURKA)
CAMK
Vidarabine
I
11
12
32
11
12
32
B
3QCQA_3Q0
(PDPK1)
CAMK
Kinome_1060
I
20
63
45
20
63
45
B
1PF8A_SU9
(CDK2)
CAMK
SU 9516
I
25
19
33
25
19
33