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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
PTK6 (
Q13882
)
Kinase group
TK
Number of conformation types
0
Number of structural templates
100 (
Total 132 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
67
2W17A_I19
(CDK2)
TK
DB07936
I
25
134
47
A
2W17A_I19
(CDK2)
TK
DB07936
I
25
134
47
25
134
47
A
3LCDA_BDY
(CSF1R)
TK
Sunitinib
I
23
168
86
23
168
86
A
3ITZA_P66
(MAPK14)
TK
P66
II
15
102
25
15
102
25
A
2IVUA_ZD6
(RET)
TK
Vandetanib
I
83
291
121
83
291
121
A
1QPDA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
2DQ7X_STU
(FYN)
TK
staurosporine
I
91
74
124
91
74
124
A
2GQGA_1N1
(ABL1)
TK
Dasatinib
I
74
32
117
74
32
117
A
1QPJA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
2HZ4A_4ST
(ABL1)
TK
staurosporine
I
159
103
156
159
103
156
A
3CKXA_STU
(STK24)
TK
staurosporine
I
176
104
141
176
104
141
A
3K54A_1N1
(BTK)
TK
Dasatinib
I
56
32
103
56
32
103
A
1SM2A_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
3OCTA_1N1
(BTK)
TK
Dasatinib
I
56
32
103
56
32
103
A
1SNUA_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1U59A_STU
(ZAP70)
TK
staurosporine
I
96
80
114
96
80
114
A
1AQ1A_STU
(CDK2)
TK
staurosporine
I
195
76
118
195
76
118
A
1XBCA_STU
(SYK)
TK
staurosporine
I
71
72
105
71
72
105
A
3A4OX_STU
(LYN)
TK
staurosporine
I
73
70
88
73
70
88
A
1BYGA_STU
(CSK)
TK
staurosporine
I
85
72
123
85
72
123
A
1XJDA_STU
(PRKCQ)
TK
staurosporine
I
121
101
106
121
101
106
A
1YVJA_4ST
(JAK3)
TK
staurosporine
I
96
90
126
96
90
126
A
1A9UA_SB2
(MAPK14)
TK
SB 203580
I
21
31
28
21
31
28
A
1PMEA_SB2
(MAPK1)
TK
SB 203580
I
16
31
26
16
31
26
A
3OBGA_SB2
(MAPK14)
TK
SB 203580
I
21
31
28
21
31
28
A
2H8HA_H8H
(SRC)
TK
Saracatinib
I
91
255
126
91
255
126
A
1PKDA_UCN
(CDK2)
TK
UCN 02
I
195
67
118
195
67
118
A
2WIHA_P48
(CDK2)
TK
VX_680
I
111
425
105
111
425
105
A
3C4DA_325
(BRAF)
TK
PLX4720
I
35
5
58
35
5
58
A
3OG7A_032
(BRAF)
TK
PLX4720
I
35
5
58
35
5
58
A
3MVLA_38P
(MAPK14)
TK
38P
I
50
308
44
50
308
44
A
3BYMA_AM0
(LCK)
TK
triazine 34
I
39
145
100
39
145
100
A
3MVMA_39P
(MAPK14)
TK
39P
I
24
247
38
24
247
38
A
3EOCA_T2A
(CDK2)
TK
5-methyl-7-p...
I
42
148
62
42
148
62
A
1YQJA_6NP
(MAPK14)
TK
AMG_706
I
19
102
43
19
102
43
A
3GENA_B43
(BTK)
TK
7-Cyclopenty...
I
29
110
67
29
110
67
A
3NUXA_3NV
(CDK6)
TK
3NV
I
8
20
21
8
20
21
A
3EIDA_PO5
(CDK2)
TK
AC1O6YZF
I
63
211
77
63
211
77
A
3C4CA_324
(BRAF)
TK
PLX4720
I
35
5
58
35
5
58
A
2IVVA_PP1
(RET)
TK
PP1
I
27
46
63
27
46
63
A
2IW8A_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
2G2HA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
1DI9A_MSQ
(MAPK14)
TK
MSQ
I
14
29
29
14
29
29
A
3RHXA_3RH
(FGFR1)
TK
6-o-tolylqui...
I
27
31
67
27
31
67
A
2IW9A_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
2HZIA_JIN
(ABL1)
TK
PD180970
I
90
77
120
90
77
120
A
3RI1A_3RH
(FGFR2)
TK
6-o-tolylqui...
I
29
33
72
29
33
72
A
3ACJA_KSS
(LCK)
TK
6,7-dimethox...
I
13
7
25
13
7
25
A
3FQSA_585
(SYK)
TK
R-406
I
64
28
102
64
28
102
A
1OZ1A_FPH
(MAPK14)
TK
4-Azaindole 6
I
18
27
28
18
27
28
A
1H1SA_4SP
(CDK2)
TK
nu6102
I
30
33
30
30
33
30
A
3ACKA_KSR
(LCK)
TK
AC1O6YMO
I
23
42
56
23
42
56
A
3IKAA_0UN
(EGFR)
TK
2jkk
I
76
120
108
76
120
108
A
3L8XA_N4D
(MAPK14)
TK
3cg2
I
91
104
65
91
104
65
A
3FKOA_FKO
(MAPK14)
TK
L-779450
I
17
7
27
17
7
27
A
1OGUA_ST8
(CDK2)
TK
ST8
I
31
21
34
31
21
34
A
3C4FA_C4F
(FGFR1)
TK
AC1O6YNE
I
23
45
56
23
45
56
A
3PIYA_585
(BTK)
TK
R-406
I
93
17
123
93
17
123
A
1QCFA_PP1
(HCK)
TK
PP1
I
31
65
68
31
65
68
A
1OIYA_N41
(CDK2)
TK
N41
I
33
49
34
33
49
34
A
1BL6A_SB6
(MAPK14)
TK
sb216995
I
46
110
50
46
110
50
A
3MDYA_LDN
(BMPR1B)
TK
LDN193189
I
12
38
42
12
38
42
A
1QPEA_PP2
(LCK)
TK
AG 1879
I
29
63
51
29
63
51
A
1OPLA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
2VTTA_LZD
(CDK2)
TK
pyrazole dia...
I
158
42
111
158
42
111
A
1WZYA_F29
(MAPK1)
TK
AC1O4W7N
I
27
48
33
27
48
33
A
2FO0A_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
2XIKA_J60
(STK25)
TK
SU11652
I
59
49
65
59
49
65
B
31
2ITYA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
B
2ITYA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITZA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITOA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
3CD3A_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
1DI8A_DTQ
(CDK2)
TK
whi-p180
I
26
68
46
26
68
46
B
2ITQA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
3LCSA_STU
(ALK)
TK
staurosporine
I
73
100
109
73
100
109
B
2ITUA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
77
287
111
B
2ITWA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
3BKBA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
1H00A_FAP
(CDK2)
TK
AC1NAE4F
I
50
94
75
50
94
75
B
2R3IA_SCF
(CDK2)
TK
2c68
I
23
89
43
23
89
43
B
2R3JA_SCJ
(CDK2)
TK
2r3j
I
27
99
49
27
99
49
B
2R3KA_SCQ
(CDK2)
TK
2r3j
I
28
95
49
28
95
49
B
2R3LA_SCW
(CDK2)
TK
2r3j
I
19
63
41
19
63
41
B
2X9FA_X9F
(EPHB4)
TK
X9F
I
46
19
86
46
19
86
B
2C68A_CT6
(CDK2)
TK
2c68
I
23
73
43
23
73
43
B
2R3RA_6SC
(CDK2)
TK
2r3j
I
13
55
30
13
55
30
B
2C69A_CT8
(CDK2)
TK
CT8
I
22
62
38
22
62
38
B
3FQEA_P5C
(SYK)
TK
AMG_706
I
24
88
63
24
88
63
B
2R3FA_SC8
(CDK2)
TK
2c68
I
22
62
43
22
62
43
B
2R3GA_SC9
(CDK2)
TK
2r3j
I
30
137
50
30
137
50
B
2XB7A_GUI
(ALK)
TK
NVP-TAE684
I
71
66
107
71
66
107
B
2VX1A_7X8
(EPHB4)
TK
DB07256
I
19
37
15
19
37
15
B
3EKNA_GS3
(INSR)
TK
pyrrolo[2,3-...
I
90
215
127
90
215
127
B
3KCKA_3KC
(JAK2)
TK
L-779450
I
13
20
44
13
20
44
B
1OIRA_HDY
(CDK2)
TK
AC1O6YZF
I
51
203
64
51
203
64
B
2C6IA_DT1
(CDK2)
TK
2c6i
I
27
41
48
27
41
48
B
2C6OA_4SP
(CDK2)
TK
nu6102
I
23
33
27
23
33
27
E
2
3G0EA_B49
(KIT)
TK
Sunitinib
I
37
40
78
E
3G0EA_B49
(KIT)
TK
Sunitinib
I
37
40
78
37
40
78
E
3G0FA_B49
(KIT)
TK
Sunitinib
I
37
40
78
37
40
78