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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
52P
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
MAPK14 (PDB code: 3HP5)
[PDB]
[PDBsum]
Inhibitor
VX-745 (HET code: 52P)
[PDB]
Summary of KIF 3HP5A_52P
(MAPK14, PDB code:
3HP5
, chain A)
Number of family interactions
42
Number of family kinase
12 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
6 (2 are BLK inhibitors)
Involved diseases
21 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
BLK and 2 inhibitors