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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
1 PRKCD related diseases
hsa04930
Type II diabetes mellitus
Summary of query kinase
Query kinase
PRKCD (
Q05655
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
95 (
Total 485 inhibitors
)
Number of PRKCD related diseases
1 (
hsa04930
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
62
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
A
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
17
127
29
A
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
41
141
45
A
2VD5A_BI8
(DMPK)
AGC
Ro 31-7549
I
19
49
12
19
49
12
A
2UV2A_GVD
(SLK)
AGC
pyrido[4,3-d...
I
21
80
62
21
80
62
A
2VN9A_GVD
(CAMK2D)
AGC
pyrido[4,3-d...
I
16
75
24
16
75
24
A
3LM0A_EBD
(STK17B)
AGC
DCL001071
I
20
106
24
20
106
24
A
3IW4A_LW4
(PRKCA)
AGC
Sotrastaurin
I
52
119
49
52
119
49
A
2OW3A_BIM
(GSK3B)
AGC
LY_333531
I
62
139
51
62
139
51
A
3EQRA_T74
(TNK2)
AGC
T74
I
34
181
86
34
181
86
A
2V7OA_DRN
(CAMK2G)
AGC
bisindolylma...
I
23
51
16
23
51
16
A
2HXLA_422
(CHEK1)
AGC
DB07075
I
15
95
36
15
95
36
A
1XJDA_STU
(PRKCQ)
AGC
staurosporine
I
121
101
106
121
101
106
A
2DQ7X_STU
(FYN)
AGC
staurosporine
I
91
74
124
91
74
124
A
2HW7A_STU
(MKNK2)
AGC
staurosporine
I
28
55
16
28
55
16
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
1Q3DA_STU
(GSK3B)
AGC
staurosporine
I
115
71
61
115
71
61
A
1BYGA_STU
(CSK)
AGC
staurosporine
I
85
72
123
85
72
123
A
1SM2A_STU
(ITK)
AGC
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
AGC
staurosporine
I
99
104
128
99
104
128
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
1U59A_STU
(ZAP70)
AGC
staurosporine
I
96
80
114
96
80
114
A
1NXKA_STU
(MAPKAPK2)
AGC
staurosporine
I
110
67
51
110
67
51
A
3CKXA_STU
(STK24)
AGC
staurosporine
I
176
104
141
176
104
141
A
2HZ4A_4ST
(ABL1)
AGC
staurosporine
I
159
103
156
159
103
156
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
2IW6A_QQ2
(CDK2)
AGC
2iw6
I
112
209
86
112
209
86
A
2WIHA_P48
(CDK2)
AGC
VX_680
I
111
425
105
111
425
105
A
1G5SA_I17
(CDK2)
AGC
H724
I
43
170
58
43
170
58
A
2HK5A_1BM
(HCK)
AGC
1BM
I
24
121
70
24
121
70
A
2F4JA_VX6
(ABL1)
AGC
VX-680
I
110
109
134
110
109
134
A
2XYNA_VX6
(ABL2)
AGC
VX-680
I
79
101
105
79
101
105
A
3E5AA_VX6
(AURKA)
AGC
VX-680
I
57
107
93
57
107
93
A
2R3NA_SCZ
(CDK2)
AGC
AC1LZZHM
I
46
175
57
46
175
57
A
2HY0A_306
(CHEK1)
AGC
AMG_706
I
23
80
49
23
80
49
A
3A2CA_PDY
(MAPKAPK2)
AGC
6-(4-methoxy...
I
32
39
21
32
39
21
A
2PZYA_B18
(MAPKAPK2)
AGC
carboline an...
I
11
56
15
11
56
15
A
3NLBA_5BE
(CHEK1)
AGC
38P
I
45
115
49
45
115
49
A
3EIDA_PO5
(CDK2)
AGC
AC1O6YZF
I
63
211
77
63
211
77
A
1YOLA_S03
(SRC)
AGC
QGPSFIYTQAON...
I
30
114
75
30
114
75
A
2J51A_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2JFLA_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
3EJ1A_5BP
(CDK2)
AGC
AC1OCFRV
I
46
92
62
46
92
62
A
2H8HA_H8H
(SRC)
AGC
Saracatinib
I
91
255
126
91
255
126
A
2BRNA_DF1
(CHEK1)
AGC
pyrrolopyrim...
I
30
119
42
30
119
42
A
2BROA_DF2
(CHEK1)
AGC
pyrrolopyrim...
I
29
109
40
29
109
40
A
3CGFA_JNF
(MAPK10)
AGC
3cgf
I
5
15
19
5
15
19
A
3PSDA_SM7
(BRAF)
AGC
pyrazole bas...
I
6
27
23
6
27
23
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
A
2JEDA_LG8
(PRKCQ)
AGC
5-Arylidene-...
I
67
19
87
67
19
87
A
2JDOA_I5S
(AKT2)
AGC
I5S
I
10
22
29
10
22
29
A
1Y57A_MPZ
(SRC)
AGC
MPZ
I
42
155
94
42
155
94
A
3EOCA_T2A
(CDK2)
AGC
5-methyl-7-p...
I
42
148
62
42
148
62
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
1ZYSA_199
(CHEK1)
AGC
2,4-Diamino-...
I
31
92
52
31
92
52
A
2BRMA_DFZ
(CHEK1)
AGC
DFZ
I
21
88
36
21
88
36
A
2VV9A_IM9
(CDK2)
AGC
2vv9
I
19
61
36
19
61
36
A
2J90A_IZA
(DAPK3)
AGC
Pyridone 6
I
40
50
42
40
50
42
A
3DDPA_RC8
(CDK2)
AGC
Roscovitine
I
42
133
57
42
133
57
A
2I40A_BLZ
(CDK2)
AGC
2i40
I
34
95
16
34
95
16
A
2HOGA_710
(CHEK1)
AGC
3-(Indol-2-y...
I
33
66
51
33
66
51
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
B
33
3KRXA_BA1
(ADRBK1)
AGC
balanol
I
14
106
29
B
3KRXA_BA1
(ADRBK1)
AGC
balanol
I
14
106
29
14
106
29
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
3BKBA_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
1WVYA_STU
(DAPK1)
AGC
staurosporine
I
83
23
55
83
23
55
B
2XCKA_MH4
(PDPK1)
AGC
MH4
I
46
431
75
46
431
75
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
1OIRA_HDY
(CDK2)
AGC
AC1O6YZF
I
51
203
64
51
203
64
B
1H07A_MFP
(CDK2)
AGC
AC1NAKJQ
I
90
241
80
90
241
80
B
2C6EA_HPM
(AURKA)
AGC
HPM
I
44
237
90
44
237
90
B
2PE2A_464
(PDPK1)
AGC
Indolinone b...
I
134
156
104
134
156
104
B
2BMCA_MPY
(AURKA)
AGC
PHA-680632
I
107
108
107
107
108
107
B
2XRUA_400
(AURKA)
AGC
VX_680
I
33
152
63
33
152
63
B
3CGOA_JNO
(MAPK10)
AGC
DB08026
I
13
32
21
13
32
21
B
2W1EA_L0E
(AURKA)
AGC
pyrazole-ben...
I
15
32
45
15
32
45
B
2R7BA_253
(PDPK1)
AGC
Kinome_3774
I
7
51
23
7
51
23
B
3COHA_83H
(AURKA)
AGC
AKI-001
I
79
88
65
79
88
65
B
3O2MA_46A
(MAPK8)
AGC
tetrazolylyp...
I
11
21
27
11
21
27
B
3NYNA_SGV
(GRK6)
AGC
SMR000127424
I
54
7
47
54
7
47
B
2VTSA_LZC
(CDK2)
AGC
DB08140
I
28
54
26
28
54
26
B
3NAYA_MP6
(PDPK1)
AGC
ZINC13474643
I
20
81
37
20
81
37
B
3QCQA_3Q0
(PDPK1)
AGC
Kinome_1060
I
20
63
45
20
63
45
B
2R3FA_SC8
(CDK2)
AGC
2c68
I
22
62
43
22
62
43
B
2R3GA_SC9
(CDK2)
AGC
2r3j
I
30
137
50
30
137
50
B
2R3IA_SCF
(CDK2)
AGC
2c68
I
23
89
43
23
89
43