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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
STK33 (
Q9BYT3
)
Kinase group
CAMK
Number of conformation types
0
Number of structural templates
48 (
Total 143 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
34
2JAMA_J60
(CAMK1G)
CAMK
SU11652
I
50
65
32
A
2JAMA_J60
(CAMK1G)
CAMK
SU11652
I
50
65
32
50
65
32
A
1AQ1A_STU
(CDK2)
CAMK
staurosporine
I
195
76
118
195
76
118
A
3CKXA_STU
(STK24)
CAMK
staurosporine
I
176
104
141
176
104
141
A
3HMOA_STU
(TTK)
CAMK
staurosporine
I
27
50
20
27
50
20
A
1NVRA_STU
(CHEK1)
CAMK
staurosporine
I
179
71
79
179
71
79
A
1NXKA_STU
(MAPKAPK2)
CAMK
staurosporine
I
110
67
51
110
67
51
A
1NVQA_UCN
(CHEK1)
CAMK
UCN 02
I
179
65
79
179
65
79
A
1PKDA_UCN
(CDK2)
CAMK
UCN 02
I
195
67
118
195
67
118
A
2VTTA_LZD
(CDK2)
CAMK
pyrazole dia...
I
158
42
111
158
42
111
A
3M2WA_L8I
(MAPKAPK2)
CAMK
Sunitinib
I
84
90
47
84
90
47
A
3H9FA_92M
(TTK)
CAMK
Mps1-IN-2
I
12
7
6
12
7
6
A
1R78A_FMD
(CDK2)
CAMK
4-alkynyl ox...
I
127
24
97
127
24
97
A
3DOGA_NNN
(CDK2)
CAMK
NSC743927
I
50
239
48
50
239
48
A
3EQPA_T95
(TNK2)
CAMK
2-aminopyrim...
I
22
92
63
22
92
63
A
3GFWA_S22
(TTK)
CAMK
1-(4-(4-(2-(...
I
21
4
18
21
4
18
A
2BROA_DF2
(CHEK1)
CAMK
pyrrolopyrim...
I
29
109
40
29
109
40
A
3DDPA_RC8
(CDK2)
CAMK
Roscovitine
I
42
133
57
42
133
57
A
3NLBA_5BE
(CHEK1)
CAMK
38P
I
45
115
49
45
115
49
A
2R3NA_SCZ
(CDK2)
CAMK
AC1LZZHM
I
46
175
57
46
175
57
A
2X9EA_SVE
(TTK)
CAMK
AZD_1152HQPA
I
3
32
5
3
32
5
A
3EJ1A_5BP
(CDK2)
CAMK
AC1OCFRV
I
46
92
62
46
92
62
A
2WMUA_ZYU
(CHEK1)
CAMK
4-(9h-purin-...
I
6
17
19
6
17
19
A
2CKEA_IQU
(DAPK2)
CAMK
AEIQS
I
10
17
22
10
17
22
A
2WU6A_DKI
(CLK3)
CAMK
5-AMINO-3-{[...
I
26
9
26
26
9
26
A
3GU8A_3GU
(DAPK1)
CAMK
Vidarabine
I
14
17
24
14
17
24
A
2HOGA_710
(CHEK1)
CAMK
3-(Indol-2-y...
I
33
66
51
33
66
51
A
1UKIA_537
(MAPK8)
CAMK
1,9-Pyrazolo...
I
20
4
24
20
4
24
A
3EIDA_PO5
(CDK2)
CAMK
AC1O6YZF
I
63
211
77
63
211
77
A
2UZBA_C75
(CDK2)
CAMK
2uzb
I
2
14
5
2
14
5
A
2ZMDA_537
(TTK)
CAMK
1,9-Pyrazolo...
I
8
4
9
8
4
9
A
2IW6A_QQ2
(CDK2)
CAMK
2iw6
I
112
209
86
112
209
86
A
2BRNA_DF1
(CHEK1)
CAMK
pyrrolopyrim...
I
30
119
42
30
119
42
A
2WIHA_P48
(CDK2)
CAMK
VX_680
I
111
425
105
111
425
105
A
1NVSA_UCM
(CHEK1)
CAMK
SB218078
I
97
6
53
97
6
53
B
14
1WVYA_STU
(DAPK1)
CAMK
staurosporine
I
83
23
55
B
1WVYA_STU
(DAPK1)
CAMK
staurosporine
I
83
23
55
83
23
55
B
1OKYA_STU
(PDPK1)
CAMK
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CAMK
UCN 02
I
179
60
109
179
60
109
B
2PE2A_464
(PDPK1)
CAMK
Indolinone b...
I
134
156
104
134
156
104
B
1UU7A_BI2
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
CAMK
bisindolylma...
I
83
189
65
83
189
65
B
1UU9A_BI3
(PDPK1)
CAMK
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
CAMK
Ro 31-7549
I
82
181
65
82
181
65
B
3ORZA_BI4
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
CAMK
bisindolylma...
I
82
178
65
82
178
65
B
1UU3A_LY4
(PDPK1)
CAMK
Ruboxistaurin
I
71
117
57
71
117
57
B
2XCKA_MH4
(PDPK1)
CAMK
MH4
I
46
431
75
46
431
75
B
2PE0A_39Z
(PDPK1)
CAMK
2pe0
I
20
2
27
20
2
27
B
1Z5MA_LI8
(PDPK1)
CAMK
BX-320
I
11
35
28
11
35
28